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3-{5-[(5-methylfuran-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-[4-(2-fluorophenoxy)phenyl]-1-propylpiperidine-4-carboxamide
2-(5-{1-[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
(4S)-3,3,4-trimethyl-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-4-ol
ethyl 4-[(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)carbamoyl]piperazine-1-carboxylate
N,1-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]-3-(pyrrolidin-1-yl)piperidine
3-(5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
N-ethyl-N-(2-hydroxyethyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
2-{1-[(dimethyl-1,3-oxazol-4-yl)methyl]-1H-1,2,3-triazol-4-yl}benzoic acid
1-[(2R,3R)-3-(dimethylamino)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(pyrazin-2-yl)propan-1-one
methyl[(3-{2-[4-(oxolane-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](1,3-thiazol-4-ylmethyl)amine
4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-1,3-dimethylpiperazin-2-one
2-{1-[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}-1,3-thiazole
(1S,5R)-6-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
[(4-ethoxyphenyl)methyl]({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
2-(2-fluorophenoxymethyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
N-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]ethane-1-sulfonamide
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydro-1-benzofuran-5-carboxamide
1-[2-methoxy-4-({[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(4-methoxyphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
4-(2,3-dihydroxypropyl)-1-(2-phenylethyl)piperazin-2-one
N-benzyl-N-methyl-3-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)methyl]imidazo[1,2-a]pyridine-2-carboxamide
3-{3-[1-(carbamoylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N-cyclopropylpropanamide
2-ethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidine-5-carboxamide
2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-1,2-dihydroisoquinolin-1-one
1-ethyl-N-(3-methoxypropyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[4-(3-methoxyphenyl)-3-oxopiperazine-1-carbonyl]benzonitrile
2-(2-aminoethyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]quinazolin-4-amine
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]propanamide
(2S,4S)-4-amino-N,N-diethyl-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidine-2-carboxamide
(1S,4S)-2-(2-methoxy-5-methylphenyl)-5-[2-(4-methylphenoxy)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(methylsulfanyl)propanamide
1-(4-cyclohexylpiperazin-1-yl)-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
3-(propan-2-yl)-5-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-yl}-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
1-cyclopentyl-4-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-one
5-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
2-(1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
5-ethyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,2-dimethylpyrimidin-4-amine
6-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyrimidin-4-amine
3-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
N,4-dimethyl-5-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
5-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]quinoxaline
2-{[(3aS,6aS)-1-(morpholine-4-carbonyl)-octahydropyrrolo[2,3-c]pyrrol-5-yl]methyl}-5-methoxy-4H-pyran-4-one
2-(dimethylamino)-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide