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3-cyclopentaneamido-N-[2-(dimethylamino)ethyl]-N-ethylbenzamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2,3-dimethylbenzamide
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methyl-N-(thiophen-3-ylmethyl)pyridin-2-amine
2-[4-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-1,4-diazepan-1-yl]-1,3-benzothiazole
1-(1'-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
(3S)-N,N-dimethyl-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}azepan-3-amine
7-[(3,4-difluorophenyl)methyl]-6-oxo-N-propyl-2,7-diazaspiro[4.5]decane-2-carboxamide
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)propanamide
5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
1-(2-{1-cyclopentyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2-methylpropyl)-4-methylpiperazine
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(9H-fluoren-9-yl)propanamide
N-[2-chloro-5-(diethylcarbamoyl)phenyl]oxolane-3-carboxamide
2-{4-[(2-fluoro-4-methoxyphenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
(3R,4R)-4-cyclopropyl-1-[(2,3-dimethoxyphenyl)methyl]-3-methylpiperidin-4-ol
1-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-propylurea
{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
N-{[3-(dimethylamino)thiolan-3-yl]methyl}-2-methyl-6-propylpyrimidin-4-amine
[(4-fluorophenyl)methyl](methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-(furan-2-ylmethyl)-1-(1H-indole-3-carbonyl)piperidine-4-carboxamide
6-(piperidin-3-yl)-2-(thiophen-3-ylmethyl)-3,4-dihydropyrimidin-4-one
2-[5-(4,5-dimethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]-2-methylpropane-1,3-diol
2-{1'-hexanoyl-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
(1R,5R)-6-(2,1,3-benzothiadiazol-5-ylmethyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-(4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperazin-1-yl)-N-(propan-2-yl)acetamide
3-(dimethyl-1,2-oxazol-4-yl)-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
1-(2-chloro-6-fluoro-3-methylbenzoyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)pyridine-3-carboxamide
1-(4-phenylbenzoyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
3-[3-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-5-(propan-2-yl)-1,2-oxazole
1-(2,6-dimethylpyridin-4-yl)-4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
{[2-(2-methylphenoxy)pyridin-3-yl]methyl}({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})amine
(1R,5R)-6-(2-methoxyethyl)-3-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
N-[(6-hydroxypyrimidin-4-yl)methyl]-4-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
2-({[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
N-methyl-3-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
N-[(3S,4R)-4-(4-methylphenyl)-1-(pyridazine-3-carbonyl)pyrrolidin-3-yl]cyclopropanecarboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
5-fluoro-N,N-dimethyl-2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]pyrimidin-4-amine
N-(5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-1-ethyl-2-(2-fluorophenyl)-1H-1,3-benzodiazol-7-yl)acetamide
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(3-hydroxyphenyl)piperidin-1-yl]propan-1-one
bis(1,3-oxazol-4-ylmethyl)({[2-(propan-2-yl)pyrimidin-4-yl]methyl})amine
4-{[5-(3-phenyl-1H-pyrazol-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]furan-2-carboxamide
8-(6-chloro-1,3-benzothiazol-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
4,6-dimethyl-2-{9-methyl-10-oxo-3,9-diazaspiro[5.6]dodecan-3-yl}pyridine-3-carbonitrile
2-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}piperidine-1-carbonyl)pyridine