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2-methoxyethyl N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carboxamide
(1-{[5-(4-cyclobutyl-6-methylpyrimidin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}piperidin-3-yl)methanol
N-[2-methoxy-5-({[1-(4-methyl-1H-imidazol-2-yl)propyl]carbamoyl}amino)phenyl]acetamide
1-(2-chlorophenyl)-2-{[2-(dimethylamino)-6-methylpyrimidin-4-yl]amino}ethan-1-ol
6-({methyl[(2-methylpyridin-4-yl)methyl]amino}methyl)pyridine-2-carboxylic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
3-chloro-N-cyclopentyl-4-({1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}oxy)benzamide
N-(3-{2-methoxy-4-[(3-methylpiperidin-1-yl)methyl]phenoxy}propyl)thiophene-2-carboxamide
5-cyclopropanecarbonyl-1'-(3-ethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(dimethyl-1,3-thiazol-5-yl)-1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
(3R,4S)-4-cyclopropyl-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]pyrrolidin-3-amine
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
N-[2-(2,4,6-trimethylphenoxy)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}pyridin-2-amine
4-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-1-methylpiperazine-2-carboxylic acid
2-[2-(1-{2-[(3-methoxyphenyl)sulfanyl]acetyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
N2,N2,N4-trimethyl-N4-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-(methylamino)-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
6-[(diethylamino)methyl]-N-(2-hydroxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[(4-{3-[4-(propan-2-yl)piperidine-1-carbonyl]piperidin-1-yl}piperidin-1-yl)methyl]pyridine
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-2-[3-(1-methoxyethyl)phenyl]pyridine
N-methyl-5-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(azepan-1-yl)-3-[3-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]methylamine
N-[2-(4-fluorophenyl)ethyl]-N-[(3-methoxyphenyl)methyl]-4-methylpyrimidine-5-carboxamide
5-ethyl-1'-[2-(methylsulfanyl)pyridine-3-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{2-oxo-2-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}imidazolidine-2,4-dione
3-({4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
(3S,4R)-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-(3-methyl-4-{[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
N-{3-[2-(2,2-diphenylethyl)morpholin-4-yl]-3-oxopropyl}acetamide
1-(1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)-2-phenylethan-1-ol
N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-(pyrazin-2-yl)-7-azaspiro[3.5]nonan-1-ol
2-methyl-1-[4-({[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)piperidin-1-yl]propan-1-one
3-chloro-1-{2-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(2-methoxyphenyl)propanamide
9-(2-amino-6-methylpyrimidin-4-yl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
(4S)-1-[2-(3-methoxyphenoxy)ethyl]-3,3,4-trimethylpiperidin-4-ol
2-(1-ethylpiperidin-4-yl)-N-[1-(4-methylpyridin-2-yl)propyl]acetamide
1-(methoxymethyl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]cyclobutane-1-carboxamide
(2S)-2-{[5-(3-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
5-(propan-2-yl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
(2S)-2-amino-N-cyclopentyl-3-methoxy-N-(3-phenylprop-2-yn-1-yl)propanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(dimethylamino)-N-methyl-2-(4-methylphenyl)acetamide
3-phenyl-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[2-(furan-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-methyl-3-phenyl-8-(quinolin-2-yl)-1,8-diazaspiro[4.5]decane