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5,6-dimethoxy-2-[(1-methylpiperidin-3-yl)methyl]-1,2-dihydroisoquinolin-1-one
1-[7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(1-methyl-1H-indol-3-yl)ethan-1-one
N-(furan-2-ylmethyl)-3-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(prop-2-en-1-yl)propanamide
1-methyl-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperazin-2-one
8-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-{4-[(4-ethylphenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-butyl-2-cyclopropyl-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-propylfuran-2-yl)methyl]piperidine
(1,4-dioxan-2-ylmethyl)({[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl})methylamine
1-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
(2S,4R)-4-amino-N,N-diethyl-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidine-2-carboxamide
1-(1-benzylpiperidin-4-yl)-N-(cyclopropylmethyl)piperidine-3-carboxamide
1,3-dimethyl-7-{2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]ethyl}-2,3,6,7-tetrahydro-1H-purine-2,6-dione
(1S,5R)-6-[(4-phenylphenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,3R)-2-amino-1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methoxybutan-1-one
N-[(5-fluoro-2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)cyclopropanamine
2-(4-chloro-1H-pyrazol-1-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}propanamide
N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-1-[(4-fluorophenyl)methyl]piperidin-3-amine
2-methyl-3-[4-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]phenol
2-methyl-4-(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)pyrimidine
3-acetamido-N-{4-[(2-methoxyethyl)carbamoyl]phenyl}pyrrolidine-1-carboxamide
(2R,3S,6R)-3-phenyl-5-(pyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(pyrrolidin-2-yl)-N-(1,2,4-triazin-3-yl)thiophene-2-carboxamide
N-cyclopropyl-1-(1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-4-yl)piperidine-3-carboxamide
(1S,6R)-9-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(2,6-difluorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{2-[4-(3-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
5-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
3-chloro-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-4-hydroxy-N-methylbenzamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(3-methoxyphenoxy)ethan-1-one
5-{2-[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]-2-oxoethyl}-1,3-dimethylimidazolidine-2,4-dione
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(1,4-dioxan-2-ylmethyl)propanamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]methylamine
1-ethyl-5-({8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1H-1,2,4-triazole
3-[(cyclopentylamino)methyl]-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
3-({6-hydroxy-4-[2-(1H-imidazol-1-yl)acetyl]-1,4-diazepan-1-yl}methyl)benzonitrile
N-cyclopropyl-4-methoxy-2-({1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}oxy)benzamide
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
3-[1-(3,5-dimethyl-1H-indole-2-carbonyl)piperidin-4-yl]phenol
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(quinolin-8-ylmethyl)piperazin-2-yl}ethan-1-ol
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidine-4-carboxylate
1-[4-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)piperidin-1-yl]ethan-1-one
3-[({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)carbamoyl]pyridin-1-ium-1-olate
7-(3-chlorophenyl)-4-(5-ethyl-1,3-oxazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[4-(1H-indol-4-yl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
(1-methoxypropan-2-yl)({[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amine
5-methanesulfonyl-2-methyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrimidin-4-amine
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-amine
4-[3-(pyridin-4-yl)-5-(pyrrolidin-3-yl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide