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N-[4-(pyridin-3-yloxy)phenyl]-1-(pyridin-4-ylmethyl)piperidine-2-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
N-[4-({methyl[3-(1H-pyrazol-1-yl)propyl]carbamoyl}methoxy)phenyl]propanamide
5-{[5-(4-methanesulfonylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-1,2,4-triazole
1,5-bis(cyclopropylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
9-[2-amino-6-(2-methylpropyl)pyrimidine-4-carbonyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
methyl 1-ethoxy-2-oxo-8-(thiophene-3-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea
1-(4-{[2-(dimethylamino)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-(thiophen-3-yl)ethan-1-one
5-(methoxymethyl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)furan-2-carboxamide
4-(5-{5-[(methylsulfanyl)methyl]furan-2-yl}-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl)pyridine
N-[(2-fluorophenyl)methyl]-3-[1-(1H-indole-6-carbonyl)piperidin-3-yl]propanamide
1-[(3-methoxyphenyl)methyl]-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
N-(adamantan-2-yl)-2-[1-(2-methoxyethyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-methyl-1H-imidazol-4-yl)methyl]benzamide
3-({1-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1,2-dihydroquinolin-2-one
1-tert-butyl-4-{[methyl({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl})amino]methyl}pyrrolidin-2-one
N,N-diethyl-1-({4-[(2-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-3-carboxamide
2-[3-methyl-4-({3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-pyrazol-1-yl]ethan-1-ol
5-(2-{8-butyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(2,3-difluoro-4-methylbenzoyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
methyl[(3-methyl-1,2-oxazol-5-yl)methyl][(2,3,4-trimethoxyphenyl)methyl]amine
N-(1-{[(2H-1,3-benzodioxol-5-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(4-fluorophenyl)-2-hydroxy-N-methylacetamide
1'-(4-propylpyrimidine-5-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-(2-aminoethyl)-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]quinazolin-4-amine
5-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-2-methoxyphenol
N-[2-(1H-pyrazol-1-yl)ethyl]-4-(pyrrolidin-3-yl)benzamide
1-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
3,5-difluoro-2-[3-(3-methoxypropyl)piperidine-1-carbonyl]pyridine
3-benzyl-4-(5-chlorofuran-2-carbonyl)piperazin-2-one
N-ethyl-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-5-carboxamide
1-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)-2-(methylsulfanyl)ethan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-1-ethyl-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}propan-1-one
N-cyclopropyl-1-[(3-fluorophenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
N-cyclopentyl-1-{1-[(3-methylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-2-phenylacetamide
1-cyclohexyl-N3,N5-dimethyl-4-oxo-N3-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}amine
2-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]pyridin-4-amine
2-(4-acetyl-1,4-diazepan-1-yl)-2-(3,4,5-trimethoxyphenyl)acetic acid
2-[(2-{1-[4-(prop-2-en-1-yl)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
4,4,4-trifluoro-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butan-1-one
4-{2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
1-ethyl-3-methyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidine-3-carboxamide
{3-[(3-chlorophenyl)methyl]-1-(5-fluoro-1H-indole-2-carbonyl)piperidin-3-yl}methanol
2-(4-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(2,2-dimethylpropyl)piperazin-2-yl)ethan-1-ol
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[3-(methylsulfanyl)propyl]amine