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(7R,9aR)-N-cyclohexyl-7-[(1S)-1-hydroxyethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-methoxypiperidine
(3R,4S)-4-[ethyl({[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl})amino]oxolan-3-ol
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyrrolidin-1-yl)pyrazine
4-(naphthalen-2-yloxy)-1-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylic acid
(4aS,7aR)-1-(2-aminopyridine-4-carbonyl)-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2,4-dimethyl-1,4-diazepane-1-carbonyl)-7-fluoro-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
1-{2-[4-(3-chloro-4-fluorophenyl)-1H-1,2,3-triazol-1-yl]ethyl}piperidine-3-carboxamide
(3S,4S)-4-[butyl(methyl)amino]-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-3-ol
5-{[(1-hydroxycyclohexyl)methyl]amino}-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-benzyl-8-(furan-3-ylmethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-[(3-methylpyridin-2-yl)methyl]propanamide
{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[(1-hydroxycyclohexyl)methyl]propanamide
(3R,4S)-4-cyclopropyl-1-[4-(difluoromethoxy)benzenesulfonyl]pyrrolidin-3-amine
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-N,N-diethylpyrrolidin-3-amine
2-hydroxy-5-(1H-pyrrol-1-yl)-N-(4H-1,2,4-triazol-4-yl)benzamide
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-{[1-(2,2-dimethylpropyl)piperidin-3-yl]methyl}quinoline-8-sulfonamide
2-cyclopropyl-8-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}oxane-4-carboxamide
2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
N-(1H-1,3-benzodiazol-2-ylmethyl)-5-(2,6-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
8-methoxy-3-[2-(morpholin-4-yl)ethyl]-3,4-dihydroquinazolin-4-one
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
methyl (2S,4S,5R)-4-(azepane-1-carbonyl)-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylate
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-(oxan-4-ylmethyl)pyridin-2-amine
7-(3-chlorophenyl)-4-[(2R)-pyrrolidine-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2E)-1-(3-{4-[(4-phenylpiperazin-1-yl)methyl]phenoxymethyl}piperidin-1-yl)-3-(thiophen-2-yl)prop-2-en-1-one
4-[3-(1H-pyrazol-3-yl)phenyl]-2-(pyrrolidin-1-yl)-6-(trifluoromethyl)pyrimidine
4-[hydroxy(pyridin-2-yl)methyl]-N-[3-(1H-1,2,4-triazol-1-yl)phenyl]piperidine-1-carboxamide
2-ethyl-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-(1-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}piperidine-4-carbonyl)morpholine
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N-(3-methoxypropyl)-1-methylpiperidin-4-amine
2-cyclopentyl-9-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-1-yl)ethyl]amine
1-(4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
6-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
1-(6-hydroxy-1,4-diazepan-1-yl)-3-[5-(thiophen-2-yl)furan-2-yl]propan-1-one
(1S,2S)-2-{[4-(ethylamino)pyrimidin-2-yl]amino}cyclohexan-1-ol
methyl 4-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}thiophene-2-carboxylate
N-[1-(2-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-{[1,2,4]triazolo[4,3-a]pyridine-7-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
4-benzyl-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-one
2-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]pyridine
4-tert-butyl-6-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-1,2-dihydropyrimidin-2-one
2-[4-(cyclopropylmethyl)-1-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
N-methyl-2-[methyl(pyridin-3-ylmethyl)amino]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-(cyclopropylmethyl)-2-(4-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}morpholin-3-yl)acetamide