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N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(1-{7-[(3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
6-(2-chlorophenyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-chloro-3-ethyl-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-methyl-1H-pyrazole
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
methyl 3-{5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}propanoate
1-(3-cyclopropylpropanoyl)-4-(4-fluoro-2-methylphenoxy)piperidine-4-carboxylic acid
2-(2-hydroxyethyl)-6-[(3-hydroxypiperidin-3-yl)methyl]-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
5-[({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
dimethyl[1-(4-{1-[(5-methyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazol-4-yl}phenyl)ethyl]amine
3-[2-(2-fluorophenyl)ethyl]piperidine
1-(4-fluorobenzoyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-(6-aminopyrimidin-4-yl)-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
3-({[2-(1H-indol-3-yl)ethyl](pyridin-3-ylmethyl)amino}methyl)pyrrolidin-3-ol
1-({[2-(furan-2-ylmethoxy)phenyl]carbamoyl}amino)cyclopentane-1-carboxamide
N-cyclobutyl-3-{[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]sulfamoyl}benzamide
N-(1-cycloheptylpiperidin-3-yl)-1-(4-fluorophenyl)cyclopropane-1-carboxamide
N-[(4-fluorophenyl)methyl]-3-[1-(1H-indole-5-carbonyl)piperidin-4-yl]propanamide
N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-N-(2,4-dimethoxyphenyl)propanamide
2-(cyclopentylmethyl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-(2-methoxyethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(1-benzylpiperidin-4-yl)methyl]-N,3,6-trimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
4-[(4-fluorophenyl)methyl]-1-(3-methoxypropyl)-3-(propan-2-yl)-1,4-diazepan-5-one
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]piperidine
N-[(5-methoxy-1H-indol-2-yl)methyl]-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-cyclopentylacetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amine
N-[3-(dimethylamino)propyl]-N-methyl-1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-amine
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-cyclopropylacetamide
1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-methyl-2-(3-methylphenoxy)butan-1-one
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2,3-dimethyl-1H-indole-7-carboxamide
2-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-5-methylpyrazine
N2-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-5-fluoro-N4-methylpyrimidine-2,4-diamine
N-(3,4-dimethylphenyl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
5-({[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}methyl)-N,N-dimethylfuran-2-carboxamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(6-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
N-cyclopropyl-N-(1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
4-[2-(4-hydroxypiperidin-1-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(2,3-dihydro-1H-indol-1-yl)-1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
N-(isoquinolin-5-ylmethyl)-N-methyl-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
4-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-1,4-oxazepan-6-ol
4-chloro-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-propanamidobenzamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-5-methylpiperidin-2-one
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)azetidine-2-carboxylic acid
2-{4-[(3-chloro-4-fluorophenyl)methyl]morpholin-3-yl}acetic acid
1-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine