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4-(4-fluorophenyl)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]butan-1-one
N-[(2,3-difluorophenyl)methyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
methyl[(5-methyl-1,2-oxazol-3-yl)methyl]{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}amine
1-ethyl-N-{2-[methyl(phenyl)amino]ethyl}-6-oxopiperidine-3-carboxamide
4-{[4-(hydroxymethyl)oxan-4-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(1-cyclohexylpiperidin-4-yl)-N-cyclopropylpiperidine-4-carboxamide
2-[methyl({4-methyl-5-[1-(1-methyl-1H-imidazole-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
N-ethyl-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
methyl 1-methyl-6-[4-(pyridin-3-yl)pyrimidin-2-yl]-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxylate
3-(4-methyl-1H-pyrazol-1-yl)-1-{2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}propan-1-one
5-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-[(3S,4R)-1-[3-(3-fluorophenyl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
5-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-(furan-2-yl)pyrimidine
2-[(2-{[2-(pyrrolidin-1-yl)ethyl]carbamoyl}phenyl)amino]acetic acid
3-(3-hydroxy-3-methylbutyl)-N-[1-(hydroxymethyl)cyclohexyl]benzamide
9-[(5-methyl-2,1,3-benzothiadiazol-4-yl)sulfonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-3-(1H-pyrazol-1-ylmethyl)benzamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[(1-methylpiperidin-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
1-[(2-chloro-4-fluorophenyl)methyl]-N-{[4-(morpholin-4-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-(2-methoxyethyl)piperidine-4-carboxamide
2-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(4-phenyl-1,2,3-thiadiazol-5-yl)pyrrolidine-1-carboxamide
1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}-3-ethylpiperidin-3-ol
N-[1-(methoxymethyl)cyclopentyl]-2-methyl-1,3-benzoxazole-6-carboxamide
1-{2-[4-(pyridin-3-yl)piperazin-1-yl]ethyl}-1H-indazole
2-(3-fluorophenyl)-N-{[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
2-methyl-5-propyl-4-(1H-pyrazol-3-yl)pyrimidine
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(naphthalen-2-yloxy)acetamide
N-(3-methylphenyl)-3-{1-[4-(1H-pyrazol-4-yl)butanoyl]piperidin-4-yl}propanamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-4-methylpentan-1-one
1-[1'-(2-ethylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
3-(4-methoxy-3,5-dimethylbenzoyl)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine
3-[(3R,4S)-1-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-(3-chloro-2,6-dimethylphenyl)-2-(2-hydroxyethyl)-3-oxopiperazine-1-carboxamide
1-cycloheptyl-5-[4-(3-methoxyphenyl)piperazine-1-carbonyl]piperidin-2-one
(3S,4R)-3-benzyl-1-[4-(hydroxymethyl)benzoyl]-4-methylpiperidin-4-ol
4-(naphthalen-1-ylmethyl)-3-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
ethyl 3-benzyl-1-[(4-acetamidophenyl)methyl]piperidine-3-carboxylate
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
2-(1-benzyl-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
3-cyclopropyl-1-methyl-5-(2-phenoxyethyl)-1H-1,2,4-triazole
2-(2-aminoethyl)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methylquinazolin-4-amine
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-methyl-2-phenylpropan-1-one
{5-[1-(3-chloro-2-methylphenyl)-1H-imidazol-2-yl]furan-2-yl}methanol
methyl 2-[8-(2,2-diphenylethyl)-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
3-(2-methoxyethyl)-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]piperidine-3-carboxylic acid
1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(oxolane-2-carbonyl)-1,4-diazepane
1'-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]