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2-(2-aminoethyl)-N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)quinazolin-4-amine
1-[2-methoxy-5-({[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
5-benzyl-3-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(4-hydroxy-3-methoxyphenyl)pyridine-3-carbonitrile
1-(2,5-dimethoxyphenyl)-3-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]urea
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[2-(4-cyclopentylphenyl)pyridine-4-carbonyl]-4-methylpiperazine
2-(4-fluorophenyl)-4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}morpholine
2-hydroxy-2-(4-methoxyphenyl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-{4-[2-(prop-2-en-1-ylsulfanyl)propanamido]phenyl}pentanamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(2-hydroxypropyl)-1H-pyrazole-4-carboxamide
2-amino-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-methyl-1,3-benzothiazole-6-carboxamide
5-{[4-(benzenesulfonyl)piperazin-1-yl]methyl}quinoxaline
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]piperidine-1-carboxamide
2-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4-methyl-1H-imidazole
5-(3-fluoro-5-methylphenyl)-4-phenyl-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-imidazole
1-(2-methoxyethyl)-8-[(3-methylquinoxalin-2-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({2-[({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]phenyl}methyl)pyrrolidin-2-one
N-[2-(azepan-1-yl)ethyl]-N-ethyl-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-4-oxo-4H-chromene-2-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]quinoline
methyl({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)[(3,4,5-trimethoxyphenyl)methyl]amine
3-(naphthalen-1-yl)-5-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]-1,2,4-oxadiazole
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[1-(thiophen-2-yl)propan-2-yl]amino}acetamide
5,6-dimethyl-N-(1-propylpiperidin-3-yl)pyrimidin-4-amine
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[(2-methyl-1H-indol-3-yl)methyl]piperidin-3-ol
N-[(5-methylthiophen-2-yl)methyl]-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
ethyl 4-(cyclopropylmethyl)-1-[3-(3-fluorophenyl)benzoyl]piperidine-4-carboxylate
(2S,4S)-4-amino-N,N-diethyl-1-[2-(2H-indazol-2-yl)acetyl]pyrrolidine-2-carboxamide
N3-(2-methoxyethyl)-N5-[(4-methylphenyl)methyl]-4-oxo-N3-(propan-2-yl)-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
9-[3-(4-fluorophenoxy)propyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(1R,2R,6S,7S)-4-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
8-methyl-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3,5-dimethylphenyl)-N'-[2-methoxy-1-(pyridin-2-yl)ethyl]-N'-methylpropanediamide
4-[2-(3-methoxyphenoxy)propanoyl]-1-(4-methylphenyl)piperazin-2-one
7-methyl-4-(3-methylphenyl)-6-(pyrimidine-4-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
2-methyl-6-[1-(quinoline-6-carbonyl)piperidin-4-yl]pyrimidin-4-ol
3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-1-{2-[2-(pyridin-2-yl)ethoxy]phenyl}urea
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(phenylcarbamoyl)ethyl]propanamide
2-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
1-butyl-4-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]piperazin-2-one
3-[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-phenyl-1,2-oxazole
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl){[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}amine
4-[1-(pyrimidin-4-yl)piperidin-4-yl]thiomorpholine
3-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
1-[2-(4-cyclohexanecarbonylpiperazin-1-yl)ethyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
N,N-dimethyl-1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}pyrrolidin-3-amine