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(3aS,6aS)-2-cyclobutanecarbonyl-5-[(2-fluoro-4-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(furan-3-yl)-1-phenyl-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-cyclopentyl-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6-oxopiperidine-3-carboxamide
9-(3-hydroxypropyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-(5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperidin-3-ol
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-(trifluoromethyl)pyridine
propan-2-yl 3-{[(2R)-2-carbamoylpyrrolidine-1-carbonyl]amino}-4-chlorobenzoate
{2-[(4aS,7aR)-6,6-dioxo-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}urea
3-[5-(4-methoxy-3-methylphenyl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
6-methyl-3-({4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}methyl)-1,2-dihydroquinolin-2-one
methyl 3-cyclohexyl-2-oxo-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
2-amino-N-{[3-(dimethylamino)phenyl]methyl}-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(2-fluoro-4-methylphenyl)-4-(3,3,3-trifluoropropyl)pyrimidine
3-(2-fluorophenyl)-N-[3-(4-methylpiperazin-1-yl)propyl]-1H-pyrazole-5-carboxamide
1'-[(2-ethylpyrimidin-4-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-[3-(1H-pyrazol-5-yl)phenyl]piperidin-4-amine
2-[2-(4-hydroxyphenyl)ethyl]-N-(trimethyl-1H-pyrazol-4-yl)piperidine-1-carboxamide
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{4-[(methoxycarbonyl)amino]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}thiomorpholine
3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]-1-(piperidin-1-yl)propan-1-one
4-chloro-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
(5-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-2-ethoxyphenyl)methanol
3-{5-[3-(1H-pyrazol-1-yl)propyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
(1S,5R)-6-(cyclopropylmethyl)-3-[4-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-methyl-6-propylpyrimidin-4-yl)-N-[(3,4,5-trifluorophenyl)methyl]piperidin-4-amine
2-cyclopropyl-3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
N-methyl-3-propyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-3-phenylprop-2-yn-1-one
methyl 1-[(3S,5S)-5-(cycloheptylcarbamoyl)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-methyl-N-[(3-methylphenyl)methyl]-4-oxo-N-(propan-2-yl)pentanamide
(3R,4R)-1-(3-chloro-5-fluorobenzoyl)-4-cyclobutyl-3-methylpiperidin-4-ol
(4aR,7aS)-1-acetyl-4-[(4-ethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
7-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
4-(2-amino-6-methylpyrimidin-4-yl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(3R,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]pyridazine-3-carboxamide
2-{[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrol-3a-yl]formamido}-N-(2,3,4-trifluorophenyl)acetamide
2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-methylpyrimidin-4-amine
3-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1-[(5-propyl-1H-pyrazol-3-yl)methyl]urea
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(2-methoxyethyl)-N-methyl-5-oxopyrrolidine-3-carboxamide
(5S,9aS,9bS)-5-[4-(difluoromethoxy)phenyl]-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-{[4-(2-hydroxyethoxy)phenyl]methyl}-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
5-{2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-1,2-oxazole-3-carboxamide