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N-(2-{[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]methyl}quinolin-6-yl)acetamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
(3S,4S)-1-[1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-4-propylpyrrolidine-3-carboxylic acid
7-fluoro-4-[3-(pyrrolidin-1-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
N-(2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1,2,3,4-tetrahydroisoquinolin-7-yl)pyridine-2-carboxamide
3-[(3R,4S)-1-[4-(2-methylpropyl)benzoyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-[(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-5-methoxy-4H-pyran-4-one
1-methyl-4-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazine
1-[(2-methoxyphenyl)methyl]-5-(thiomorpholine-4-carbonyl)piperidin-2-one
3-{[1-(3-hydroxybenzoyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-[2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrimidin-4-yl]piperidin-4-ol
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
3-[1-(5-aminopyridin-3-yl)-1H-1,3-benzodiazol-2-yl]propan-1-ol
N4-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-6-methylpyrimidine-2,4-diamine
(4aR,8aS)-6-(4-fluorobenzoyl)-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N4-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-5-butyl-6-methylpyrimidine-2,4-diamine
7-(1,3-benzothiazol-2-yl)-4-cyclopropanecarbonyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-[(2,6-dimethylphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-[2-(1H-pyrazol-1-yl)phenyl]-1,4-diazepane-1-carboxamide
N-{[1-ethyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-fluoro-3-methylbenzene-1-sulfonamide
N-[(3-methylpyridin-2-yl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
2-[1-(2,3-dimethylphenyl)-5-[5-(1H-pyrazol-1-ylmethyl)furan-2-yl]-1H-1,2,4-triazol-3-yl]acetamide
{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
5-[2-(pyridin-3-yl)-1H-imidazol-1-yl]pyridin-2-ol
1-[5-(4-chloro-2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-cyclohexylpiperazine
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-methylbenzamide
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidin-2-amine
3-[1-(1-benzylpiperidin-4-yl)piperidin-4-yl]-N-cyclopropylpropanamide
N-(cyclohexylmethyl)-3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
4-(1-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}piperidine-4-carbonyl)morpholine
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-5-propyl-1,2-oxazole-4-carboxamide
3-(1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-3-carbonyl)pyridine
2-ethoxy-5-[4-phenyl-1-(pyridin-3-ylmethyl)-1H-imidazol-5-yl]pyridine
N,N,4,5-tetramethyl-6-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}pyrimidin-2-amine
1-{1-[(3-phenyloxolan-3-yl)methyl]azetidin-3-yl}piperidine
4,6-dimethyl-3-{4-[(1-methylpiperidin-3-yl)methyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
1-[3-(2-fluorophenoxy)azetidin-1-yl]-3-(1-methylpiperidin-2-yl)propan-1-one
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-3-(2-hydroxyphenyl)propan-1-one
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2,4-dimethyl-1,3-thiazole-5-carboxamide
5-fluoro-2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
5-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
2,5-dimethyl-N-[(5-methylfuran-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-benzyl-1-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-cyclopentyl-4-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperazine
{4-fluoro-7-[6-(trifluoromethyl)pyridin-3-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
1-(3-methoxyphenyl)-3-methyl-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazin-2-one
(3aR,6aR)-2-(cyclobutylmethyl)-5-(4-methylpyridine-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid