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3-(2-methoxyphenyl)-N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}propanamide
1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-(3-fluoro-4-methylphenyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
methyl 4-[(5-methanesulfonamido-2-methylphenyl)carbamoyl]piperazine-1-carboxylate
N-[2-(4-methoxyphenyl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(5-phenyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-yl]methanol
4,6-dimethyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
8-hexanoyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[4-(1H-pyrazol-1-yl)butan-2-yl]amine
2-(2-fluorophenyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-methyl-4-{1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}piperidin-4-ol
3-chloro-N-[2-(dimethylamino)ethyl]-4-[(1-ethylpiperidin-4-yl)oxy]benzamide
3-ethyl-N-[2-(4-methoxyphenyl)ethyl]-1-methyl-N-[(1-methylpiperidin-4-yl)methyl]-1H-pyrazole-5-carboxamide
4-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl}benzoic acid
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(propan-2-yl)pyrimidin-2-amine
2-(ethylamino)-N,4-dimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1,3-thiazole-5-carboxamide
1'-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-[(3R,4S)-1-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
ethyl 4-[(3-methoxyphenyl)methyl]-1-(3-phenylprop-2-yn-1-yl)piperidine-4-carboxylate
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-methylpiperidin-2-one
3-(1H-1,3-benzodiazol-1-yl)-1-[3-(3-methoxyphenoxy)azetidin-1-yl]propan-1-one
5-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methoxyphenol
N-[3-(1H-imidazol-1-yl)propyl]-1-methyl-5-oxo-N-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(1,3-dimethyl-1H-pyrazol-5-yl)-1H-pyrazol-1-yl]acetamide
1-{4-[(2,3-dihydroxypropyl)(methyl)amino]pyrimidin-2-yl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-cyclopropyl-9-[(3,4-dimethylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
{1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
2-{1'-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
(2E)-N-[2-(3-acetamidophenyl)phenyl]but-2-enamide
methyl 3-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-9-[(1-methylpiperidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
4-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-oxobutane-1-sulfonamide
N-(5-{[(1R,5S,8R)-8-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}pyrimidin-2-yl)benzenesulfonamide
3-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
1-[2-(4-methoxyphenyl)ethyl]-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}piperidin-2-one
6-[(dimethylamino)methyl]-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrimidin-4-amine
3-{imidazo[1,2-a]pyridin-2-yl}-1-(4-methyl-1,4-diazepan-1-yl)propan-1-one
methyl 3-(2-methoxybenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
ethyl 4-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)piperazine-1-carboxylate
N-benzyl-1-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-ethylpiperidine-3-carboxamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,8-naphthyridine
2-({3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-4-methoxyphenol
3-phenyl-N-(4-{4-[(prop-2-en-1-yl)amino]piperidin-1-yl}phenyl)propanamide
2-[({1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}oxy)methyl]pyridine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-(1H-imidazol-1-ylmethyl)furan-2-carboxamide
3-[2-(2,2-diphenylethyl)morpholine-4-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
methyl 2-{2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methylacetamido}acetate