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5-methoxy-3-[(4-phenyl-1,3-thiazol-5-yl)methyl]-3,4-dihydroquinazolin-4-one
4-(3-methylthiophene-2-carbonyl)-7-(pyrrolidin-1-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(furan-2-carbonyl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-1,4-diazepane
2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methylacetamide
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methylpiperidine
1-(2H-1,3-benzodioxole-5-carbonyl)-4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
7-[(3-methoxyphenyl)methyl]-2-(1-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
5-propyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,2-oxazole-3-carboxamide
3-fluoro-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
6-[(2-fluorophenyl)methoxy]-4-(5-methyl-1,2-oxazole-3-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
2-(morpholin-4-ylmethyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-1,4-oxazepane
1-[(6-ethoxyquinolin-2-yl)methyl]-2-methyl-1,4-diazepan-5-one
1-{4-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]phenyl}ethan-1-one
1-{2-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
(3S,5R)-5-(cyclopropylcarbamoyl)-1-(2,3-dichlorobenzoyl)piperidine-3-carboxylic acid
2-(5-acetylthiophen-3-yl)-N-[(3,5-difluorophenyl)methyl]acetamide
4-(1H-1,3-benzodiazole-5-carbonyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-methoxy-1-(4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N'-{2-[(pyridin-3-yl)amino]ethyl}-N-(2,4,6-trimethylphenyl)butanediamide
N-{[3-(methylsulfanyl)phenyl]methyl}-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3,3,3-trifluoropropanamide
5-({3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)-2-methoxyphenol
7-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
1-(3-methylbutyl)-8-(oxan-4-yl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(pyridin-4-ylmethyl)-4-{[1-(1,3-thiazol-2-yl)piperidin-4-yl]oxy}benzamide
N-[(5-chlorothiophen-2-yl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
6-(3-methoxyphenyl)-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[(2E)-3-(furan-2-yl)prop-2-en-1-yl](oxolan-2-ylmethyl)amine
(1R,2S)-N1-tert-butyl-N2-{3-[(pyridin-3-yl)amino]propyl}cyclohexane-1,2-dicarboxamide
N-(1,3-benzothiazol-6-yl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-3-(2-methylphenyl)pyrrolidin-3-ol
N-(1-benzothiophen-5-ylmethyl)-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
1-(2-propylpyridine-4-carbonyl)-4-(pyrrolidine-1-sulfonyl)piperazine
(3S)-3-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)azepan-2-one
2-hydroxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
methyl 7-oxo-9-(pyridin-2-ylmethoxy)-3-(2,4,5-trifluorobenzoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[4-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
ethyl 1-[(6-methylpyridin-2-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
6-[1-(4-methoxyphenyl)cyclopropyl]-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-9H-purin-2-amine
4-[(2,3-difluorophenyl)methyl]-3-{2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
4-(propan-2-yl)-6-[3-(pyrrolidin-1-yl)pyrrolidin-1-yl]pyrimidine
{[5-(4-chloro-2-fluorophenyl)furan-2-yl]methyl}[2-(1H-imidazol-4-yl)ethyl]amine
4-{3-[(3-chlorophenyl)methyl]-5-(1H-imidazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
1-(2-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
5-(3-acetylphenoxymethyl)-N-cyclopentyl-1H-pyrazole-3-carboxamide
2-(4-{4-[3-(methoxymethyl)piperidin-1-yl]piperidin-1-yl}benzoyl)-1,2,3,4-tetrahydroisoquinoline