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N-(1,2-oxazol-3-ylmethyl)-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-3-methyl-N-(2-methylpropyl)furan-2-carboxamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
(4aS,8aR)-6-(3-methylfuran-2-carbonyl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
ethyl 1-(2-methylpyridine-3-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
6-[ethyl(methyl)amino]-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
3-hydroxy-S-[2-(pyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]butane-1-sulfonamido
2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
N5-benzyl-N3-methyl-4-oxo-N3-(2-phenylethyl)-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-methyl-4-{[(3-phenyl-1H-pyrazol-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
1'-(3-ethyl-1,2-oxazole-5-carbonyl)-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(4-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}phenyl)-1H-pyrazole
3-hydroxy-3-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-(piperazin-1-yl)ethan-1-one
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
2-{[6-(thiomorpholin-4-yl)pyrazin-2-yl]sulfanyl}acetic acid
9-methoxy-7-(pyridin-3-yl)-4-[4-(trifluoromethoxy)benzenesulfonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(2-amino-1,3-thiazol-4-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
9-[(5-hydroxy-2-methoxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-3-(2-oxooxolan-3-yl)propanamide
N-(2-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-oxoethyl)acetamide
methyl 4-(4-{1-[(4-fluorophenyl)methyl]-4-methyl-2,5-dioxoimidazolidin-4-yl}piperidine-1-carbonyl)benzoate
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-3-(propan-2-yl)-1,2-oxazole
5-methyl-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indazole
8-(4-chloro-2-fluorobenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-cyclopropyl-9-[(4-methyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-2-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}quinoline
N-(butan-2-yl)-2-(2-methylphenoxy)-N-(pyridin-4-ylmethyl)acetamide
3-[1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-2-yl]pyridine
4-(2,2-dimethylpropyl)-3-{2-oxo-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethyl}piperazin-2-one
methyl 2-{8-[1-(methylsulfanyl)propan-2-yl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
4-(benzyloxy)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]butan-1-one
methyl 5-oxo-5-(4-{2-[(pyridin-3-ylmethyl)carbamoyl]ethyl}piperidin-1-yl)pentanoate
3-(azocan-1-yl)-1-[4-(6-methylpyridin-2-yl)piperazin-1-yl]propan-1-one
2-{4-[(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}pyrimidine
N-[(1R)-1-(4-chlorophenyl)ethyl]-5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
3-[({[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}amino)methyl]piperidin-3-ol
2-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-1,2-dihydroisoquinolin-1-one
4-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-oxobutanamide
1-[(4aR,8aS)-1-[2-(2-methylphenyl)acetyl]-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
N-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-7-methoxy-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-{[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
1-(2-ethoxypyridine-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-benzyl-4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
6-[4-(2,3-dihydro-1H-indene-1-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
N-[2-({[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}amino)ethyl]methanesulfonamide
4-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](benzyl)amino}butan-1-ol
2-{2-[(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
2-(pyrrolidin-1-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
ethyl 1-[2-(4-methoxyphenyl)ethyl]-5-(5-methylpyrazine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate