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N-(2-methylpropyl)-1-[1-(3-phenylpropanoyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetamide
3-benzyl-8-{[2-(furan-2-yl)phenyl]methyl}-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-1-[(2E)-4-methylpent-2-en-1-yl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
methyl 4-({[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]amino}methyl)benzoate
8-[(4-hydroxyphenyl)methyl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(adamantan-1-yl)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]ethan-1-one
2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-{1-ethyl-5-[(1R,2R)-2-phenylcyclopropanecarbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-phenylpiperazine
(2S)-N2-[2-(3-methoxy-4-propoxyphenyl)ethyl]pyrrolidine-1,2-dicarboxamide
8-methoxy-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-methylpyrimidin-2-amine
3,3-dimethyl-1-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
2-{4-[2-(2,5-dimethoxyphenyl)acetyl]morpholin-3-yl}acetamide
N-(dimethyl-1H-1,2,4-triazol-3-yl)-3-propoxypiperidine-1-carboxamide
1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
1-(3,4-dimethylphenyl)-N-[(2-methoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(dimethylamino)-N-[(2-ethoxypyridin-3-yl)methyl]-2-(2-fluorophenyl)acetamide
3-[(dimethylamino)methyl]-1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-3-ol
2-(3-methoxyphenyl)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)pyrrolidine-1-carboxamide
3-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
4,4,4-trifluoro-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}butan-1-one
1-[(3-fluorophenyl)methyl]-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
N-[2-(4-{[4-(4-chlorophenyl)butanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]oxolane-2-carboxamide
2-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
N,N-dimethyl-5-[1-(propan-2-yl)piperidine-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
4-{3-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-1,3-thiazol-2-amine
2-[(4-methoxyphenyl)methyl]-4-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
(3R,4R)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
2-{4-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-1-yl}-1,3-benzoxazole
2-{2-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-oxoethyl}-4-phenyl-1,2-dihydrophthalazin-1-one
7-(cyclobutylmethyl)-2-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane
5-ethyl-7-{octahydro-1H-pyrido[1,2-a]piperazin-2-yl}pyrazolo[1,5-a]pyrimidine
3-chloro-N-cyclopentyl-4-({1-[1-(pyridin-2-yl)propan-2-yl]piperidin-4-yl}oxy)benzamide
3-(3-methoxyphenyl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
[(3R,4R)-1-(2-chloro-4-fluorobenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1,9-dimethyl-10-oxo-N-[4-(propan-2-yl)phenyl]-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)amine
2-[(4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazin-1-yl)methyl]benzonitrile
3-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,3-dichlorophenyl)urea
8-benzyl-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(4-fluoro-2-methylphenyl)-2-{[3-(oxolan-3-yl)propyl]amino}acetamide
5-(1H-1,3-benzodiazole-5-carbonyl)-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-amino-4-{2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
3,3-dimethyl-4-[6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carbonyl]piperazin-2-one