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(3R,5R)-1-benzyl-N-(oxolan-2-ylmethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(pyridin-3-yl)propanamide
3-(3-fluorophenyl)-4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperazin-2-one
N,N-dimethyl-5-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-1,3-thiazol-2-amine
4-(2-fluoro-5-methylphenoxy)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
1-cyclohexyl-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
4-{2-[2-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-5-oxopyrrolidin-1-yl]ethyl}benzene-1-sulfonamide
(2S,4S,5R)-4-[(furan-3-ylmethyl)carbamoyl]-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
2-cyclopentyl-8-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[5.5]undecan-3-one
1-(4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
4-(1-benzofuran-3-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-6-oxo-1-(prop-2-en-1-yl)piperidine-3-carboxamide
butyl N-[(3R,5S)-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}pyrrolidin-3-yl]carbamate
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
2-[methyl(piperidin-4-yl)amino]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
7-[2-(2-amino-4-methyl-1,3-thiazol-5-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-(2-chlorophenyl)-N-(4-hydroxybutyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]acetamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-(2-ethoxyethyl)-5-(morpholine-4-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-2-methylphenol
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(thiophen-2-yl)ethan-1-one
N,N,4-trimethyl-3-{[(5-methylpyridin-3-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
methyl (2S)-1-{5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carbonyl}pyrrolidine-2-carboxylate
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
(2R)-2-amino-3-(4-chlorophenyl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]propan-1-one
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
(3R,4S)-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-propylpyrrolidin-3-amine
(1R,2S)-N1-(prop-2-en-1-yl)-N2-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]cyclohexane-1,2-dicarboxamide
1-acetyl-N-[(3R,4S)-1-(2-hydroxyethyl)-4-phenylpyrrolidin-3-yl]piperidine-4-carboxamide
3-chloro-N-[(2-ethoxypyridin-3-yl)methyl]-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
8-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[1-(3-phenylpropyl)-5-(thiophen-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
N-methyl-1-[(2-methylphenyl)methyl]-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
N-(1-{7-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
N-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
2-[4-(2-methoxyphenyl)-1H-pyrazol-1-yl]-N-[1-(pentan-2-yl)-1H-pyrazol-5-yl]acetamide
(3aS,6aS)-1-oxo-5-(3-phenyl-1,2,4-oxadiazol-5-yl)-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[(1-benzylpyrrolidin-3-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
5-fluoro-2-(4-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
[3-(2-methoxyethyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-3-yl]methanol
2-(4-ethylpiperazine-1-carbonyl)-4-(thiophen-3-ylmethyl)morpholine
1-(carbamoylmethyl)-N-[1-(2,5-difluorophenyl)cyclopropyl]piperidine-4-carboxamide
3-methoxy-5-{thieno[2,3-d]pyrimidin-4-yl}pyridine
N-cyclobutyl-5-(2,4-difluorophenoxymethyl)-1H-pyrazole-3-carboxamide
6-{[3-(4-carboxyphenyl)piperidin-1-yl]methyl}pyridine-2-carboxylic acid
{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
3-[3-(1-methoxyethyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid