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methyl 4-(4-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-(2-methylphenyl)-2-{[5-(phenoxymethyl)-1H-pyrazol-3-yl]formamido}acetamide
3-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-4H-chromen-4-one
6-methyl-5-{5-[(2,5,7-trimethyl-1H-indol-3-yl)methyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
1-(3,5-dimethylphenyl)-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazin-2-one
4-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-(thian-4-yl)piperazine
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[4-(methylsulfanyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
7-(1,3-benzothiazol-2-yl)-4-benzyl-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-(2,3-dihydro-1H-inden-2-yl)-1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane
N4-[1-(2-phenylethyl)piperidin-3-yl]pyrimidine-4,6-diamine
2-(4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)pyridine-3-carbonitrile
[1-(4-methoxy-3-methylbenzoyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
2-(4-benzoylpiperidin-1-yl)-4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyrimidine
1-[(4aS,8aS)-4a-hydroxy-7-(1H-imidazol-2-ylmethyl)-decahydro-2,7-naphthyridin-2-yl]-2-methoxy-2-methylpropan-1-one
1-[(2-chlorophenyl)methyl]-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
(2S)-2-{[7-(cyclopropylmethyl)-6-(4-methoxyphenyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}propanamide
6-(4-fluorophenyl)-N-(2-hydroxyethyl)-N-methyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[3-(2-methoxybenzamido)phenyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyrrolidine-1-carbonyl)pyridine
2-({9-oxo-1-oxa-8-azaspiro[4.6]undecan-8-yl}methyl)benzonitrile
1-(2-hydroxy-3-methoxybenzoyl)-3-(hydroxymethyl)piperidin-3-ol
2-amino-6-(3-methylphenyl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[1-phenyl-3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}amine
(1S,5R)-3-(1,3-benzothiazol-2-yl)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
2-(4-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)propanoic acid
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
2-methyl-4-{3-[2-(pyridin-2-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
N-(2-chlorophenyl)-3-[1-(1,3-thiazol-2-yl)piperidin-4-yl]propanamide
1-cyclopropyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-oxopyrrolidine-3-carboxamide
3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-{[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-ethyl-1-[(4-ethynylphenyl)methyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
N-[(2R,3R)-2-methoxy-1'-(quinolin-5-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N-(oxolan-2-ylmethyl)-4-{[2-(1H-pyrazol-4-yl)ethyl]sulfamoyl}benzamide
1-phenyl-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}butane-1,4-dione
1-(3-methylbutyl)-3-(pyrimidin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
2-[({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(propan-2-yl)amino]ethan-1-ol
1-(2,3-dihydro-1H-inden-2-yl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(5-methylpyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(5S,9aS,9bS)-5-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2,5-dimethyl-3-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
1-[3-(dimethylsulfamoyl)-5-{[(2-fluoro-5-methoxyphenyl)methyl]amino}benzoyl]piperidine-3-carboxamide
(2R)-2-hydroxy-2-phenyl-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one