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N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-ethylbutanamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-1-ethyl-N-methyl-1H-pyrazole-4-carboxamide
3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
3-({[1-(oxolan-3-ylmethyl)piperidin-4-yl]oxy}methyl)pyridine
1-methyl-3-(5-methylpyridin-3-yl)-1-(oxan-2-ylmethyl)urea
(3R,5S)-1-benzyl-N-[(3,4-difluorophenyl)methyl]-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-3-amine
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]acetamide
3-(3-methoxyphenoxy)-1-(2-propoxybenzoyl)azetidine
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(2,3-dimethoxyphenyl)methyl]pyrrolidine-2-carboxylate
N-{1-[4-(dimethylamino)phenyl]propan-2-yl}-4-methylpiperidine-4-carboxamide
5-methyl-3-(3-phenylpropyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
5-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-phenyl-1H-imidazole-4-carboxamide
4-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-2,1,3-benzoxadiazole
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
(3S,5R)-1-(3-methoxypropanoyl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
1-(5-tert-butyl-2-methoxyphenyl)-3-ethyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
(3S,4R)-1-({3-carboxypyrazolo[1,5-a]pyrimidin-6-yl}methyl)-4-phenylpyrrolidine-3-carboxylic acid
benzyl(methyl){[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}amine
N,5,7-trimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
3-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-5-(3,4-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
3-(2-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
(3aR,5S,6S,7aS)-2-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-octahydro-1H-isoindole-5,6-diol
1-(1-benzofuran-3-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-(4-fluorophenoxy)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidine
N-(1-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-butyl-5-chloro-2-oxo-N-(thiophen-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
5-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
(2S)-2-(methoxymethyl)-N-(1-phenyl-1H-pyrazol-5-yl)pyrrolidine-1-carboxamide
2-[5-(methoxymethyl)-4-(2-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
2-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
{5-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]furan-2-yl}methanol
5-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)propan-1-one
2-amino-4-[4-(dimethylamino)phenyl]-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-(azocan-1-yl)-3-(5-{[(3-ethoxypropyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
4-({[(3-chloro-4,5-diethoxyphenyl)methyl]amino}methyl)-1,2-dihydrophthalazin-1-one
N-[2-(ethylsulfanyl)ethyl]-4-hydroxy-2-phenylpyrimidine-5-carboxamide
N-(2-methoxyethyl)-N-methyl-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
1-(2-methoxyphenyl)-3-(1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]acetamide
2,5-dimethoxy-N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
(2S)-N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-5-oxopyrrolidine-2-carboxamide
{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}dimethylamine
N-methyl-N-(1-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}-2-phenylethyl)thiophene-2-carboxamide
N-[2-(2,5-dimethylphenoxy)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
4-chloro-3-fluoro-N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}benzamide
(3R,5R)-5-(pyrrolidine-1-carbonyl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide