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methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(2-methoxyacetamido)-5-[(2-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-3,4-dihydroquinazolin-4-one
2-[3-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenyl]-6-(3-methylpyrazin-2-yl)-3,4-dihydropyrimidin-4-one
N-[1-(4-methoxyphenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-5-methyl-1,2-oxazole-3-carboxamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-{[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}pyrrolidine-2-carboxamide
[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]({[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})methylamine
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(morpholine-4-sulfonyl)-2-(3-phenylpropyl)morpholine
N-(2-methyl-1-benzofuran-5-yl)-4-(2-methylpyrimidin-4-yl)piperidine-1-carboxamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
1-[(3,4-dimethoxyphenyl)methyl]-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
5-[methyl({[1-(piperidin-1-yl)cyclohexyl]methyl})carbamoyl]-1H-imidazole-4-carboxylic acid
4-(2-fluoro-4-methylbenzoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
{5-[(2-benzylmorpholin-4-yl)methyl]furan-2-yl}methanol
1-methyl-8-{[1-(propan-2-yl)-1,2,3,4-tetrahydroquinolin-6-yl]methyl}-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-4-(2-methoxyphenyl)-1-(3-propyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
2-(morpholin-3-yl)-N-(thiophen-2-ylmethyl)acetamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
2-({[4-(methylsulfanyl)phenyl]methyl}({[3-(pyrimidin-2-yloxy)phenyl]methyl})amino)ethan-1-ol
5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(1H-pyrazol-4-yl)pyridine
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
{2-[(6-chloropyridin-2-yl)oxy]hex-5-en-1-yl}(methyl)(pyridin-3-ylmethyl)amine
1-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-3-[4-(methylsulfanyl)benzoyl]piperidine
4-[(5-ethylpyridin-2-yl)methyl]-9-(furan-2-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecane
4-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]piperidine-1-sulfonamide
N-methyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
5-[4-(furan-2-ylmethyl)piperazine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
3-[(cyclopropylamino)methyl]-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
2,5-dioxo-6-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-({[5-(4-chloro-2-fluorophenyl)furan-2-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl]amino)ethan-1-ol
N-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]benzamide
3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-5,6,7,8-tetrahydroquinoline
1-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-cyclopentyl-3-[5-(3-methoxypropanoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
3-(2-methylpropyl)-1-(2-phenylethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(3-ethyl-3-hydroxypiperidin-1-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
2-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,2-oxazinane
8-{[6-(dimethylamino)pyridin-3-yl]methyl}-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1-{[3-(morpholin-4-yl)phenyl]methyl}-3-propylpiperidin-3-yl)methanol
1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(4-methylphenyl)ethan-1-one
N-[1-(2-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-oxoethyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
(1S,5R)-6-benzyl-3-[2-(morpholin-4-yl)-2-oxoethyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(3,4-dichlorophenyl)piperazin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-hydroxy-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methylbenzamide
6,8-dimethyl-2-({[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]amino}methyl)quinolin-4-ol
8-(butan-2-yl)-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
benzyl(cyclopropylmethyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
5-cyclobutanecarbonyl-1'-(oxane-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]