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N-(propan-2-yl)-2-(pyridin-3-yloxy)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-(quinoxalin-2-ylmethyl)benzamide
2-[4-(2-fluoro-4-methylbenzoyl)morpholin-3-yl]acetic acid
{[5-(oxan-2-yl)furan-2-yl]methyl}(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
3-[(1-ethyl-1H-1,3-benzodiazol-2-yl)sulfanyl]-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]propan-1-one
N'-(adamantan-1-yl)-N-[2-(dimethylamino)ethyl]-N-methylpropanediamide
1-[2-(4-fluorophenyl)morpholin-4-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
ethyl 4-(3-cyano-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridin-6-yl)piperidine-1-carboxylate
N-[(2R,3R)-1'-[(2-hydroxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
N-[(3R,5S)-1-(1,4-dithiepan-6-yl)-5-(methylcarbamoyl)pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
butyl (4aS,7aR)-6,6-dioxo-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
2-[(4,4-difluoropiperidin-1-yl)methyl]-8-methoxyquinoline
N-[1-(morpholin-4-ylmethyl)cyclopentyl]-4-propylpyrimidine-5-carboxamide
2-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-ol
2-(4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
8-(3-ethyl-1,2-oxazole-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
2-methyl-1-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)-1,4-diazepan-5-one
(3S,4R)-4-(2-methylphenyl)-1-[2-(pyrrolidin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
2-cyclopropyl-4-phenyl-9-(piperidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-phenylethyl)-6-(pyridin-4-ylmethoxy)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
2-methyl-4-{3-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
2-(1-propylpiperidin-4-yl)-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]ethan-1-one
1-{3-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
N-({3-[7-(5-ethylpyrimidin-2-yl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
3-(2-methoxyethyl)-1-[(3-methoxyphenyl)methyl]-5-methyl-1H-1,2,4-triazole
6-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
6-(4-cyclopentylpiperazin-1-yl)-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(4-phenylbutyl)propanamide
2-({[5-(methoxymethyl)furan-2-yl]formamido}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-4-methyl-N-(2-methylpropyl)-1,2,5-oxadiazole-3-carboxamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(2-methyl-1H-indol-3-yl)ethyl]acetamide
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)acetamide
2-[(5-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}pyridin-2-yl)amino]acetamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(3-hydroxy-3-methylbutyl)-N-methyl-1,3-oxazole-4-carboxamide
4-(5-methylpyridin-2-yl)-1-(4-phenoxybutyl)piperidin-4-ol
(3R,4R)-1-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
1-ethyl-N-[(2-{3-[2-(4-methoxyphenyl)acetamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
2-(dimethylamino)-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,4-dimethylpyrimidine-5-carboxamide
(3R,4R)-4-amino-1-({2-[4-(1H-imidazol-1-yl)butoxy]phenyl}methyl)piperidin-3-ol
2-(dimethyl-1,3-thiazol-5-yl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
6-(1H-indol-6-ylmethyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
[1-(2,3-difluoro-4-methoxybenzoyl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
N-[(2-fluorophenyl)methyl]-1-methyl-5-(4-propylpiperazin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(3-hydroxypropyl)-9-(2-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-benzyl-5-[(4-methyl-1H-imidazol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-(piperidin-3-yl)benzamide
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(2-methylpropyl)carbamoyl]pyrrolidine-2-carboxylic acid
2-{4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}pyrimidine