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3-({[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amino}methyl)-4H-chromen-4-one
{3-[(4-fluorophenyl)methyl]-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl}methanol
(2R,3R,6R)-3-(4-fluorophenyl)-5-(1H-imidazol-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{5-[(2,6-difluorophenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-1H-pyrazole
1-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pentane-1,2-dione
4-[(4-{[1-(thiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]morpholine
4-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-1H-pyrrole-2-carbonitrile
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidine
N-(3,4-dimethoxyphenyl)-1-[2-(2-fluorophenyl)benzoyl]piperidin-3-amine
N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyl-1-(pyridin-2-yl)piperidine-3-carboxamide
2-(cyclopropylmethyl)-9-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
[(5-chlorofuran-2-yl)methyl](methyl)[2-(oxan-4-yl)ethyl]amine
1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(4-fluorophenyl)methyl]-3-[1-(thiophene-2-carbonyl)piperidin-4-yl]propanamide
methyl (2S)-2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-3-(4-hydroxyphenyl)propanoate
2-{[(4aS,8aR)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]methyl}benzoic acid
(4aS,8aR)-1-(2-methylpropyl)-6-(2-propylpyridine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
2-[4-(cyclohexylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
3-(1H-1,3-benzodiazol-2-ylmethyl)-5-methoxy-3,4-dihydroquinazolin-4-one
1-(4-{[4-(difluoromethoxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-phenylethan-1-ol
N-methyl-N-[1-(pyridin-3-yl)ethyl]-2-(pyridin-4-ylsulfanyl)acetamide
6-ethyl-2-methyl-4-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}quinoline
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-cyclopropyl-N-({4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)-4-(morpholin-4-yl)benzamide
2-(5-{1-[5-(carboxymethyl)pyrimidin-4-yl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-[2-(trifluoromethyl)benzoyl]-6-azaspiro[2.5]octane
2-[5-(5-chloro-6-oxo-1,6-dihydropyridin-3-yl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
4-methyl-N-{2-methyl-5-[3-(1,2-oxazinan-2-yl)propanamido]phenyl}benzamide
1-(3-fluorophenyl)-3-{1-[1-(4-formylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
7,11-dimethyl-3-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3,7,11-triazaspiro[5.6]dodecane
4-({[(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amino}methyl)-N-methylbenzene-1-sulfonamide
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(4-ethoxyphenyl)ethan-1-one
(1R,5R)-6-(cyclobutylmethyl)-3-(2-fluoro-4-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
4-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
4-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}thiomorpholine
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
(2S,4S)-4-amino-N-methyl-1-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)pyrrolidine-2-carboxamide
N-(3,3-diphenylpropyl)-6-[(2-hydroxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(azepane-1-carbonyl)phenyl]-1H-1,2,4-triazole-5-carboxamide
2-[(cyclopropylmethyl)sulfanyl]-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-{4-[(2-chloro-4-fluorophenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{3-methyl-5-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)phenyl]-1H-1,2,4-triazol-1-yl}pyridine
(2R,6S)-2,6-dimethyl-N-[4-(thiophen-2-ylmethoxy)phenyl]morpholine-4-carboxamide
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]({[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2-methyl-5-{pyrazolo[1,5-a]pyridin-7-yl}-1,3-benzothiazole
4-[(2-fluorophenyl)methyl]-3-(furan-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{1-[2-(4-methylphenoxy)acetyl]piperidin-4-yl}-N-phenylpropanamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol