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2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}acetamide
N-[(2R,3R)-1'-[(4-hydroxy-3,5-dimethylphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
2-methyl-4-[4-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)phenyl]but-3-yn-2-ol
N-(4-{2-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-1H-imidazol-1-yl}phenyl)acetamide
1-{5-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-4-phenylbenzamide
2-methanesulfonamido-N-methyl-N-(thiophen-3-ylmethyl)propanamide
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-4-(piperidin-3-yl)benzamide
methyl 4-[2-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)ethyl]piperidine-1-carboxylate
3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]urea
1-cyclohexyl-5-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(5-chloro-2-ethoxyphenyl)-6-fluorobenzamide
1-methyl-4-(2-{1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperidin-2-yl}ethyl)piperazine
1-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
N,3,5-trimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-benzofuran-2-carboxamide
(2R,3R)-3-amino-1'-(quinolin-4-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine
5-{1-[4-(1H-indol-3-yl)butan-2-yl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
N-ethyl-2-(4-fluorophenyl)-N-[(5-methylfuran-2-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
2-{[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]methyl}-6-methylquinolin-4-ol
2-amino-3-ethyl-N-[(1-hydroxycyclohexyl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
6-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-(4-methyl-1,4-diazepane-1-carbonyl)-6-azaspiro[2.5]octane
4-{5-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
1-{4-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-2-(1H-imidazol-4-yl)ethan-1-one
2-hydroxy-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
2-(2-methoxyethyl)-8-[(1-methyl-1H-indol-6-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-phenyl-N-(1-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
5-[1-(3-methyl-2-oxopentanoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N-[2-(morpholin-4-yl)ethyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
N-(4-acetylphenyl)-3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxypyridine-4-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)benzamide
2-[3-(azepan-1-ylmethyl)-6-chloroimidazo[1,2-a]pyridine-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
8-fluoro-2-(3,3,3-trifluoropropyl)-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
2-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(3,4-dimethylphenyl)-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[(2-methyl-1H-indol-5-yl)methyl]acetamide
(1r,4r)-4-({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)cyclohexan-1-ol
2-(cyclohex-1-en-1-yl)-N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}acetamide
2-hydroxy-1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
6-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}pyridine-2-carboxylic acid
3-[5-(2,5-dimethylphenyl)-6-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl]-1-methylpyrrolidin-2-one
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-2-methylpropan-1-one
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-4-yl)propanamide
2-[4-benzyl-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
4-[2-(2-methoxyphenoxy)-2-methylpropanoyl]-1-phenylpiperazin-2-one
3-(2-methoxyphenyl)-4-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,6-difluorobenzamide