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2-[(3-chlorophenyl)methyl]-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
6-[2-(1-methylpiperidin-2-yl)ethyl]-5,6-dihydro-1,6-naphthyridin-5-one
6-(2-hydroxyethyl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(1,4-dithiepan-6-yl)-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
(1R,3s,6r,8S)-4-[6-(piperidin-3-yl)pyrimidin-4-yl]-4-azatricyclo[4.3.1.13,8]undecane
4-(4-{[4-(propan-2-yl)phenyl]methyl}piperazin-1-yl)-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
5-({methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
1-{[5-(methoxymethyl)furan-2-yl]methyl}-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-(2-ethoxyethyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-(furan-2-yl)-2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethane-1,2-dione
5-(2,4-difluorophenoxymethyl)-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2-oxazole-3-carboxamide
4-[(3,5-dimethoxyphenyl)methyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(oxolan-3-ylmethyl)piperazine
[4-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenyl]methanol
N-[3-(1H-indol-2-yl)phenyl]-1-(pent-4-enoyl)piperidine-3-carboxamide
2-ethyl-8-[6-(4-methylpiperazine-1-carbonyl)pyrazin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]ethan-1-one
N,N-dimethyl-2-{[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-{[1-(3-methylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}acetamide
3-(4-methoxyphenyl)-N-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
4-chloro-1-methyl-3-{[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-indazole
3-[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-2H-chromen-2-one
2-{2-[(4-cyclohexyl-1,4-diazepan-1-yl)methyl]phenoxy}ethan-1-ol
1-[7-(1,3-benzothiazol-2-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
2-methyl-4-{3-[2-(pyridin-3-yl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
1,3,6-trimethyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(4-{1-[5-(ethanesulfonyl)-2-hydroxyphenyl]-1H-imidazol-2-yl}phenyl)acetamide
6-{[(1-methoxypropan-2-yl)amino]methyl}-2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)-3,4-dihydropyrimidin-4-one
3-cyano-N-(1-phenylbutyl)benzamide
(5S)-4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,2,2,5-tetramethylpiperazine
(4aS,8aR)-6-(2-hydroxyacetyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
8-fluoro-N-methyl-4-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,4-dihydroquinoline-3-carboxamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidine-3-carboxylate
methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}){[3-(trifluoromethyl)phenyl]methyl}amine
3-({[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
4-(2,6-dimethylpyridin-3-yl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]pyrimidin-2-amine
N-({1-[(2-cyanophenyl)methyl]piperidin-3-yl}methyl)propane-1-sulfonamide
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
1-(4-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}thiophen-2-yl)ethan-1-one
5-{1-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}pyrimidine
(4aS,8aR)-6-(4-methyl-1H-imidazole-2-carbonyl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-(2,5-difluorobenzoyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[(5-{[2-(3-fluorophenyl)piperidin-1-yl]methyl}pyrimidin-2-yl)(methyl)amino]acetic acid
N-[1-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-4-methyl-1-oxopentan-2-yl]thiophene-2-carboxamide
4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-5-methyl-2-phenyl-1H-imidazole
N,N-bis(prop-2-en-1-yl)-2-[4-(pyrimidin-2-yloxy)piperidin-1-yl]acetamide
1'-{[5-(oxan-2-yl)furan-2-yl]methyl}-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{[2-(dimethylamino)ethyl](methyl)amino}-2-[4-(methylsulfanyl)phenyl]acetic acid
5,6-dimethyl-2-[2-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-(azepane-1-sulfonyl)-5-(2-carboxyphenyl)benzoic acid