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4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-phenylethyl)piperidine
2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)-N-[(1s,4s)-4-aminocyclohexyl]acetamide
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S,4R)-4-amino-1-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}-N-methylpyrrolidine-2-carboxamide
1-{1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-[2-(3,4-dimethoxyphenyl)ethyl]-4-[3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N-cyclohexyl-N-methylacetamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(1H-1,2,4-triazol-5-ylmethyl)benzamide
2-amino-1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-methylpropan-1-one
4-({2-[2-(5-methylfuran-2-yl)phenyl]-1H-imidazol-1-yl}methyl)pyrimidine
N-(furan-2-ylmethyl)-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(thiophen-3-yl)acetamide
N-[(5-chloro-1H-indol-2-yl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-methyl-N-(2-methylpropyl)acetamide
N-ethyl-2-(4-fluorophenyl)-N-(oxolan-2-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
3-{[(4aS,7aR)-4-(2-hydroxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
N-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-4-yl)methanesulfonamide
4-[4-({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)piperidin-1-yl]-N-(pyridin-3-ylmethyl)benzamide
N6-cyclopropyl-N4-[3-(dimethylamino)propyl]-N4-methylpyrimidine-2,4,6-triamine
(3S,4S)-1-[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-yl]-4-(propan-2-yloxy)pyrrolidin-3-ol
methyl 3-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)propanoate
3-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,5,6-trimethyl-1,2-dihydropyridin-2-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-(4-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
2-(2-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-2-azaspiro[4.4]nonan-3-one
1-[1-(2-methylpyridin-4-yl)piperidin-4-yl]piperidin-4-ol
1-(2-hydroxyethyl)-5-(1-methylpiperidine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
2-amino-4-(3-ethyl-1H-pyrazol-5-yl)-6-(propan-2-yl)pyridine-3-carbonitrile
N-(2-{1-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}quinolin-6-yl)acetamide
1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
1-(4-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
(4aR,8aR)-7-{[3-(difluoromethoxy)phenyl]methyl}-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
2-methyl-N-({5-[(2-phenoxyethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)propanamide
N-[2-(2-fluorophenyl)-1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
(4aR,8aR)-6-[(2E)-3-phenylprop-2-en-1-yl]-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-decahydro-1,6-naphthyridine
2-[(3-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]carbamoyl}phenyl)amino]acetic acid
3,5-dimethyl-1-(1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}azetidin-3-yl)-1H-pyrazole
2-(4-propanoylphenoxy)-N-[1-(thiophen-2-yl)propan-2-yl]acetamide
2-amino-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-methylpropanamide
2-{2-[1-(3-chlorothiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-[(2,6-difluoro-3-methylphenyl)methyl]-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
N-methyl-N-[2-methyl-3-(pyrrolidin-1-yl)propyl]-3-phenylcyclobutan-1-amine
5-(2-{2-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)ethyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
[1-(4-methoxybenzenesulfonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
1-[1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]-3-methylbutan-1-one
2-(cyclopropylmethyl)-9-(2-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-[3-(1H-1,3-benzodiazol-2-yl)azetidine-1-carbonyl]-4-methyl-1,3-thiazol-2-amine