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2-{[(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)oxy]methyl}pyridine
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-7-oxo-2-(pyridine-4-amido)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-(3-hydroxy-3-phenylpropyl)-1-methyl-3-[2-(piperidin-1-ylmethyl)phenyl]urea
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-[1-(pyridin-2-yl)propan-2-yl]piperidin-4-amine
5-(2-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)-1H-1,2,3,4-tetrazole
3-(1-methyl-1H-imidazole-2-carbonyl)-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}oxolane-3-carboxamide
3-methyl-7-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
methyl 2-(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)(4-phenylbutan-2-yl)amine
5-methyl-1-{2-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
8-(2,4-dimethylpyrimidine-5-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
6-[(2-methyl-1,3-thiazol-5-yl)methyl]-1-propyl-3-[4-(1H-pyrazol-1-yl)phenyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-(2-methoxyethyl)-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[cyclohexyl(methyl)amino]-3-[3-(morpholin-4-ylmethyl)phenoxy]propan-2-ol
1-[(5-chloro-1-benzothiophen-3-yl)methyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
{4-[(3-fluorophenyl)methyl]-1-(pyrazin-2-yl)piperidin-4-yl}methanol
1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
2-(dimethylamino)-4-methyl-N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]pyrimidine-5-carboxamide
N-cyclopropyl-1-[1-(3-ethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
3-cyclopentyl-N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)propanamide
6-[(3,5-dimethoxyphenyl)methoxy]-4-(1H-indole-5-carbonyl)-1-(propan-2-yl)-1,4-diazepan-2-one
9-cyclopropanecarbonyl-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3-phenylprop-2-ynamide
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[2-(3-methylpyridin-2-yl)ethyl]benzamide
3-({4-[1-(furan-3-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
1-[4-({[2-(2-methylphenoxy)pyridin-3-yl]methyl}amino)piperidin-1-yl]ethan-1-one
N-[2-(3-methoxyphenyl)ethyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-(propan-2-yl)acetamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)(methyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
(1-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl)methanamine
(1S,5R)-6-(2-methoxyethyl)-3-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(3-methoxyphenyl)methyl]pyrrolidin-3-yl]methanol
3-methyl-1-(1-{6-[methyl(prop-2-en-1-yl)amino]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
N-({1-[2-(pyrazin-2-yl)acetyl]piperidin-3-yl}methyl)-1H-indazole-3-carboxamide
(2E)-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-[(4-hydroxyphenyl)methyl]acetamide
3-methyl-1-[(3-methylphenyl)methyl]-4-[3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanoyl]piperazin-2-one
2-[4-(2,3-dihydro-1-benzofuran-5-carbonyl)morpholin-3-yl]-1-(4-methylpiperidin-1-yl)ethan-1-one
N-{[1-(2,5-dimethylbenzenesulfonyl)piperidin-3-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
(2S)-2-{3-[(2-methoxyphenyl)methyl]-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl}pyrrolidine-1-carboxamide
2-(4-fluorophenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]imidazo[1,2-a]pyridine-6-carboxamide
5-chloro-2-fluoro-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]benzamide
4-(thiophen-2-ylmethyl)-N-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]piperazine-1-carboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide