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methyl 3-(furan-2-amido)-1-(2-methoxyethyl)-5-[(2-phenylethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-3-methyl-5-propyl-1-benzofuran-2-carboxamide
1-(3-ethoxybenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
5-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
N-(furan-2-ylmethyl)-1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]piperidine-4-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[(1R,2S)-2-phenylcyclopropyl]-2-propyl-1,3-thiazole-4-carboxamide
5-(1-{9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carbonyl}pyrrolidin-2-yl)thiophene-2-carboxamide
6-chloro-3-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amino}methyl)-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
N-[(5-fluoro-2-methylphenyl)methyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
1-[(1-{6-[2-(hydroxymethyl)phenyl]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(1S,4S)-2-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-2-azabicyclo[2.2.1]heptane
1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(5-methyl-1,2-oxazol-3-yl)piperidine
N-phenyl-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}morpholine-2-carboxamide
4-(1-benzyl-1H-imidazol-2-yl)-1-(oxolane-2-carbonyl)piperidine
2-(2-ethyl-1H-imidazol-1-yl)-1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}ethan-1-one
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
1-(3-aminoazepan-1-yl)-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
7-(3-chlorophenyl)-4-(6-methylpyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-N-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}piperidine-1-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[2-(4-methyl-2-oxo-1,2-dihydroquinolin-1-yl)acetyl]piperidin-3-yl]propanoic acid
N-(2-methoxyethyl)-2,5-dimethyl-N-(propan-2-yl)-1,3-thiazole-4-carboxamide
4-(1-hydroxy-2-{4-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}ethyl)phenol
7-(5-chloropyridin-2-yl)-4-(quinoxalin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2-methoxyethyl)-4,6-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[(4-methanesulfonylmorpholin-2-yl)methyl]amino}acetamide
1-ethyl-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
ethyl 4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine-1-carboxylate
6-methyl-2-[3-(pyridin-2-yl)azetidin-1-yl]pyridine-3-carboxamide
N-[(4-fluorophenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[3-(2-methoxybenzamido)phenyl]-4-methyl-1,2,5-oxadiazole-3-carboxamide
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amine
1-ethyl-N-{3-[methyl(phenyl)amino]propyl}-1H-pyrazole-5-carboxamide
N-({1-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)acetyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
3-(but-2-yn-1-yl)-5-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
N-[(4-chlorophenyl)methyl]-N-(3-hydroxypropyl)-1,7-dimethyl-1H-indole-2-carboxamide
4-[3-(benzyloxy)piperidine-1-carbonyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-3-yl]methyl}-2-(2-methoxyphenoxy)acetamide
1-(furan-2-ylmethyl)-N-[2-(5-methylfuran-2-yl)ethyl]piperidine-3-carboxamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(diethylamino)ethan-1-one
1-(3-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]methyl}phenyl)ethan-1-one
5-chloro-3-[1-(pyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
4-({5-[(benzyloxy)methyl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
5-[bis(prop-2-en-1-yl)amino]-1-(cyclohexylmethyl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(1-cyclopentyl-4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
N-(3,4-difluorophenyl)-1-(1H-pyrazol-3-ylmethyl)piperidin-3-amine
N-{1-oxa-8-azaspiro[4.5]decan-3-yl}-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide