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2-hydroxy-4-methyl-1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}pentan-1-one
2-cyclopropyl-4-hydroxy-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}pyrimidine-5-carboxamide
6-[1-(4-chloro-2-methylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N-({7-[2-(3-chlorophenoxy)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
N-{1-[1-(2-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-phenylethyl)piperidine
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
(4aR,8aS)-6-(1H-pyrrol-2-ylmethyl)-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
(3S)-N,N-dimethyl-1-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}azepan-3-amine
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-4-(1H-pyrazol-1-yl)benzamide
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
2-chloro-N-[2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]benzamide
(2S,4R)-4-[3-(2-amino-1,3-thiazol-4-yl)propanamido]-1-(furan-3-ylmethyl)-N-methylpyrrolidine-2-carboxamide
1-(3,3-dimethyl-2-oxobutyl)-5-oxopyrrolidine-3-carboxylic acid
2-(2-amino-6-methylpyridin-3-yl)-6-methoxy-N,N-bis(propan-2-yl)benzamide
1-[4-(1H-pyrazol-4-yl)butanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
[(3-fluorophenyl)methyl]({[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)(pyrimidin-4-ylmethyl)amine
N-[2-(1H-indol-1-yl)ethyl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
2-[4-(2-methoxyethoxy)phenyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
N-cyclohexyl-1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-3-carboxamide
3-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetic acid
2-(dimethylamino)-4-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}pyrimidine-5-carboxamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(2-{1-benzyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenoxy)acetamide
3-[3-(3-chlorobenzoyl)piperidine-1-carbonyl]-N,N-dimethylaniline
N-({5-[(4-ethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
(3R,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine
2-methyl-4-[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]-6-(piperidin-4-yl)pyrimidine
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-2-(2-methoxyphenyl)pyrimidine
5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-2-(thiophen-2-yl)pyrimidin-4-ol
1-[(4aS,8aS)-7-(5-acetylthiophene-2-carbonyl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
6-(2-fluorophenyl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(3R,4S)-4-cyclopropyl-1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]pyrrolidin-3-amine
6-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pyridine-3-carboxamide
N-(1-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2-methyl-1,3-thiazole-4-carboxamide
4-methoxy-4-phenyl-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidine
methyl (2S,4R)-4-(4-fluorobenzamido)-1-[(4-fluorophenyl)methyl]pyrrolidine-2-carboxylate
(4aS,7aR)-1-(2-methylpyrimidine-5-carbonyl)-4-pentanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-methyl-1,2-oxazol-5-yl)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
8-[(3-chloro-4-methoxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl (2S,4R)-1-[(4-methoxy-3-methylphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
1-(3,5-dimethylphenyl)-N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
6-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
1-(cyclopropylmethyl)-N-methyl-5-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-[(dimethylamino)methyl]piperidin-4-ol