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2-cyclopropyl-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(oxolan-2-ylmethyl)-9-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-fluoro-4-methoxy-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
5-(2,3-dihydro-1H-indene-1-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-cyclopentyl-3-[5-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
[(3R,5R)-1-(3-propyl-1H-pyrazole-4-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-ethenyl-N-methyl-1H-pyrazole-4-carboxamide
5-ethyl-N-[3-(4-methylpiperazin-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(4,6-dimethylquinolin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]ethan-1-one
2-methyl-5-phenyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
(1S,9R)-11-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[2-(2-methylphenyl)ethyl]carbamoyl}pyrrolidine-2-carboxylate
1-[3-(3-cyclopentyl-1,2,4-oxadiazol-5-yl)propyl]pyrrolidin-2-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-sulfonamide
1-(pyridin-3-ylmethyl)-N-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-3-amine
3-(azepane-1-carbonyl)-N-[2-(morpholin-4-yl)ethyl]-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-cyclopropyl-2-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
(2S,4S)-4-amino-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3,3,3-trifluoropropan-1-one
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
methyl (2S)-3-methyl-2-{[1-(4,6,7-trimethylquinazolin-2-yl)piperidin-4-yl]formamido}butanoate
methyl 4-[2-amino-3-cyano-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
N-butyl-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
5-(hydroxymethyl)-2-methyl-4-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)pyridin-3-ol
4-{[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]methyl}-5-tert-butylfuran-2-carboxamide
3-[2-(2-methoxyphenoxy)phenyl]-1-methyl-1-(oxan-2-ylmethyl)urea
2-{4-[(8-fluoroquinolin-2-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
3-(3-methylbutyl)-8-(4-methylpyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 4-{[4-(cyclohexylamino)quinazolin-2-yl]methyl}piperazine-1-carboxylate
2-(methylsulfanyl)-5-[4-(2-phenoxyethyl)piperazine-1-carbonyl]pyrimidine
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-3-(1-methylpiperidin-2-yl)propanamide
2-{5-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl}acetic acid
3-[(2-amino-5-ethylpyrimidin-4-yl)amino]-N-cyclohexylpropanamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidine
4-(3-fluorophenyl)-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
N-({1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
4-[(3-methyl-1,2-oxazol-5-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]ethan-1-one
3-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-N-(2,4-dimethoxyphenyl)propanamide
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
8-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(4aS,7aR)-1-(1-methylcyclopropanecarbonyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(piperidin-4-yl)-2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)-3,4-dihydropyrimidin-4-one
2-(dimethylamino)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide