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1-{4-[(5-hydroxy-4,4-dimethylpentyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-[4-(1-cyano-1-methylethyl)phenyl]-2-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}acetic acid
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-(1,3-thiazole-5-carbonyl)-6-azaspiro[2.5]octane
[(dimethyl-1,2-oxazol-4-yl)methyl][(3-ethyl-1,2-oxazol-5-yl)methyl]methylamine
benzyl({[6-chloro-4-(morpholin-4-yl)quinazolin-2-yl]methyl})ethylamine
4-(3-methylbutyl)-3-{2-oxo-2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
(3aR,6aR)-N-[3-(2-methoxyphenyl)propyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
3-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]-1-ethyl-6-methyl-1,2-dihydropyridin-2-one
N4-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
6-(4-cyclopentylphenyl)-2-methyl-2,3-dihydropyridazin-3-one
6-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-2-methyl-1,3-benzoxazole
N-ethyl-2-[3-(1-methoxyethyl)phenyl]pyridine-4-carboxamide
2-{[5-(phenoxymethyl)-1H-pyrazol-3-yl]formamido}-N-(propan-2-yl)acetamide
3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydroquinolin-2-one
7-(naphthalen-1-ylmethyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
8-(1,3-benzothiazol-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(4-cyclobutyl-6-methylpyrimidin-2-yl)phenol
N-[2-(2-chloro-6-methylphenoxy)ethyl]-5-oxopyrrolidine-3-carboxamide
N-[2-(1,3-benzothiazol-2-yl)ethyl]-4-sulfamoylbenzamide
2-cyclopentyl-9-(2-ethylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(thiophen-3-ylmethyl)benzamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
2-methyl-8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[4.5]decan-3-one
N-(4-cyclohexylphenyl)-3-oxopiperazine-1-carboxamide
1-(4-butylbenzenesulfonyl)-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
4-{[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
3-{5-[(5-methyl-1H-pyrazol-1-yl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
1-(1-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)ethan-1-one
[(1-cyclopentylpiperidin-3-yl)methyl][(6-methylpyridin-2-yl)methyl][2-(piperidin-1-yl)ethyl]amine
1-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
(3R,4R)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3,4-dimethylpyrrolidin-3-ol
N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(2-methylphenyl)-3-phenylpropanamide
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
4-{[3-(2-{4-[3-(4-fluorophenyl)benzoyl]piperazin-1-yl}ethoxy)phenyl]methyl}morpholine
2-(1-{[3-(pyridin-2-yl)phenyl]methyl}pyrrolidin-2-yl)pyridine
5-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-hydroxypiperidin-4-yl]-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
4-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}phenol
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-ol
N-{[7-chloro-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
2-[2-(3-methoxyphenyl)ethyl]-4-[3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
7-[(2-methoxyphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[4-(8-methoxyquinolin-2-yl)-1H-pyrazol-1-yl]acetamide
N-[2-(morpholin-4-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
N-ethyl-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carboxamide
1-(4-chlorophenyl)-2-[(5,6-dimethylpyrimidin-4-yl)amino]ethan-1-ol
6-[4-fluoro-2-(trifluoromethyl)phenyl]-N-methylpyridine-2-carboxamide
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})(pyridin-2-ylmethyl)amine
(4aS,7aR)-1-[(3-acetyl-2,4,6-trimethylphenyl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione