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(1S,4S)-2-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)-2-azabicyclo[2.2.1]heptane
[1-(4-fluorophenyl)propyl]({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
4-{1-[(3-chloro-4-ethoxyphenyl)methyl]piperidin-4-yl}pyridine
N-(2,3-dimethylphenyl)-2-oxo-2-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}acetamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)formamido]-2-(2-fluorophenyl)acetic acid
N-[1-(pyridin-3-yl)propan-2-yl]-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
5-(2,6-difluorophenoxymethyl)-N-[(5-methylthiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
2-({2-amino-6-[4-(4-methylphenoxy)piperidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
4-[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepane-1-carbaldehyde
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
3-(3-hydroxyquinoxalin-2-yl)-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]propan-1-one
1-(4-{[(3-ethoxypropyl)amino]methyl}-2-methoxyphenoxy)-3-(4-ethylpiperazin-1-yl)propan-2-ol
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-phenoxypropan-1-one
4-(1H-imidazol-2-ylmethyl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
3,5-dimethoxy-N-{[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]methyl}benzamide
2-(1,4-dimethylpiperazin-2-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
N-{3-[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]phenyl}methanesulfonamide
4-(1-ethyl-1H-imidazol-2-yl)-1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidine
N-methyl-5-[(methylsulfanyl)methyl]-N-[(1-phenylpyrrolidin-3-yl)methyl]furan-2-carboxamide
4-(pyridin-3-yl)-2-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]pyrimidine
4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1-(3-methylphenyl)-1H-pyrazole
7-(2-cyclohexylethyl)-2-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-2,7-diazaspiro[4.5]decane
4-benzyl-3-{1-[4-(methylamino)pyrimidin-2-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
[(2-fluorophenyl)methyl](2-methoxyethyl)(1,3-thiazol-2-ylmethyl)amine
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-(4-methyl-1H-pyrazol-1-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
3-chloro-N-[4-(4-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
5-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
2-(cyclopropylmethyl)-9-[2-(4-fluorophenyl)-2-hydroxyacetyl]-2,9-diazaspiro[5.5]undecan-3-one
1-({3-[4-(propan-2-yl)piperidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-1,3-benzodiazole
1-{1-[6-(4-methoxypiperidin-1-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
1-[(2-fluorophenyl)methyl]-N-methyl-N-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-3-amine
N-cyclopentyl-N-[2-(dimethylamino)ethyl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
N-{[2-(2-methoxypyridin-3-yl)phenyl]methyl}propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-ol
2-({[5-(hydroxymethyl)furan-2-yl]methyl}(pyridin-3-ylmethyl)amino)butan-1-ol
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
5-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-chloro-1,2-dihydropyridin-2-one
9-(3,5-difluoropyridine-2-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
4-{[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(pyrazin-2-yl)propanamide
3-{[(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
N-[4-({4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenyl]acetamide
3-[({4-benzyl-5-[1-(cyclohexylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)methyl]pyridine
1-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-4-ol
N-cyclopropyl-N-[(4-ethylphenyl)methyl]-4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(2-{1-[(3,5-difluoro-4-methoxyphenyl)methyl]piperidin-2-yl}ethyl)acetamide
dimethyl[2-(4-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}morpholin-2-yl)ethyl]amine
2-[methyl(phenyl)amino]-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide