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3-({2-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]acetamido}methyl)-4-methylbenzoic acid
N-[2-(benzyloxy)ethyl]-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-7-fluoro-3-methyl-1H-indole
(2-methylpropyl)({[5-(oxan-2-yl)furan-2-yl]methyl})(pyridin-2-ylmethyl)amine
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]pyridine-2-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-5-methyl-4-[(thiophen-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-[(1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidin-4-yl)methyl]acetamide
3-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
2-amino-N-(2-hydroxyethyl)-4-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-1,3-thiazole-5-carboxamide
(3aR,6aR)-2-(oxan-4-yl)-5-(pyridazine-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(6-hydroxy-4-methyl-1,4-diazepan-1-yl)-6-phenylpyridine-3-carboxylic acid
1-{4-[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]butan-2-yl}-4-methylpiperazine
methyl 5-{[(2,3-dimethoxyphenyl)methyl]amino}-3-(furan-2-amido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[1-(1-benzylpiperidin-4-yl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
methyl 3-ethyl-2-(furan-3-yl)-3H-imidazo[4,5-b]pyridine-6-carboxylate
N-(2,3-dihydro-1H-inden-2-yl)-4-hydroxy-N-propyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]-N-[(1S,2R)-2-phenylcyclopropyl]piperidine-1-carboxamide
N-[(2,5-difluorophenyl)methyl]-3-ethyl-4-methyl-1,2-oxazol-5-amine
2-(2,4-difluorophenyl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
N-{1-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
3-{[1-(1,3-dihydroxypropan-2-yl)pyrrolidin-3-yl]methyl}benzamide
3-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(morpholin-4-yl)ethyl]acetamide
3-cyclopropyl-1-(2,2,2-trifluoroethyl)-5-(2,4,5-trimethoxyphenyl)-1H-1,2,4-triazole
1-(3-chlorophenyl)-4-[2-(3-methoxyphenyl)acetyl]piperazin-2-one
2-{4-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]piperazin-1-yl}pyrazine
8-methoxy-5-{5-methylthieno[2,3-d]pyrimidin-4-yl}quinoline
2-(5-ethyl-1-benzofuran-3-yl)-1-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}ethan-1-one
N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,4-dithiepan-6-amine
N,2,5-trimethyl-1-phenyl-N-[1-(pyridin-3-yl)propyl]-1H-pyrrole-3-carboxamide
({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)[1-(1H-pyrazol-1-yl)propan-2-yl]amine
1-{5-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
4-[1-(5-amino-4-phenyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]pyrimidin-2-amine
N-(oxolan-3-yl)-3-phenylbenzamide
N-cyclopropyl-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-[(3-methylthiophen-2-yl)methyl]acetamide
3-[1-(furan-2-carbonyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-{1-cyclopentyl-4-[(4-methoxy-2,5-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)methanol
(4aS,8aR)-1-(2-aminoethyl)-6-(quinoline-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-methyl-7-[2-(3-phenylpyrrolidin-1-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-1-[(3-fluorophenyl)methyl]piperazin-2-one
3-hydroxy-1-(2-methoxyethyl)-3-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)piperidin-2-one
2-(2,5-dimethyl-1H-pyrrol-1-yl)-5-acetamido-N-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]benzamide
(1S,3R)-N,2,2,3-tetramethyl-3-(1-methyl-1H-1,2,4-triazol-5-yl)cyclopentane-1-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-(1-methyl-1H-pyrazole-4-carbonyl)piperazin-2-one
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
3-[2-(azetidin-1-yl)-2-oxoethyl]-2-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-4-one
4-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
2-(1H-imidazol-2-yl)-N-(1-methanesulfonylpiperidin-4-yl)benzamide