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2,2-diphenyl-1-[4-(thian-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
1-(4-fluorophenyl)-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]cyclopropane-1-carboxamide
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
5-oxo-1-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}pyrrolidine-3-carboxylic acid
(2S,4R)-4-amino-1-{2-[(2,3-dimethylphenyl)carbamoyl]acetyl}-N-ethylpyrrolidine-2-carboxamide
N-{1-oxa-8-azaspiro[4.5]decan-3-yl}-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
2-cyclopentyl-9-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-4-amine
1-cyclobutanecarbonyl-N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]piperidine-4-carboxamide
N,3-dimethyl-N-(oxan-4-yl)-5-propyl-1-benzofuran-2-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-(3-cyanopiperidin-1-yl)pyridine-3-carboxamide
1-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}azepan-2-one
methyl 4-[5-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
2-(3-chlorophenyl)-1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-imidazole
2-{1-cyclopentyl-4-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(adamantan-1-yl)-4-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperazine
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-{4-[(dimethylcarbamoyl)amino]phenyl}-4-methoxy-N-methylbenzamide
N-[1-(1-cyclopentylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxy-2-phenylacetamide
6-{[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]methyl}naphthalen-2-ol
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
4-(1,2-benzothiazol-3-yl)-N-(1,3-dihydro-2-benzofuran-5-yl)piperazine-1-carboxamide
2-(5-fluoro-2-methoxyphenyl)-1-[2-methoxy-2-(thiophen-2-yl)ethyl]-1H-imidazole
[(3-ethyl-1,2-oxazol-5-yl)methyl]({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl})methylamine
4-({2-[1-(3-fluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(dimethylamino)-N-ethyl-2-(3-methylphenyl)-N-(oxan-4-ylmethyl)acetamide
methyl 3-[7-chloro-2-({pyrazolo[1,5-a]pyrimidin-2-ylformamido}methyl)-2,3-dihydro-1-benzofuran-5-yl]benzoate
1-{2-oxo-2-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethyl}-1,2-dihydropyrimidin-2-one
1-[(2-butyl-1H-imidazol-4-yl)methyl]-8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decane
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}acetamide
4-{2-[3-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)phenoxy]ethyl}morpholine
1,3-dimethyl-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(5-fluoropyridin-2-yl)-6-methoxy-N,N-bis(propan-2-yl)benzamide
1-{[3-(difluoromethoxy)phenyl]methyl}-3-(3-methoxyphenoxy)azetidine
N-(2H-1,3-benzodioxol-5-yl)-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-3-(pyrazin-2-yl)-N-(pyridin-3-ylmethyl)propanamide
methyl(pyrazin-2-ylmethyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
3,4-difluoro-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl}ethan-1-ol
ethyl 1-[(2-methoxy-5-methylphenyl)carbamoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(1H-indazol-1-yl)acetamide
(3S)-1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-ol
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}acetamide
2-(ethylamino)-4-methyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1,3-thiazole-5-carboxamide
3-(prop-2-en-1-yl)-1-(pyridin-4-yl)piperidine-3-carboxylic acid
(3S,4S)-1-[(2-fluoro-5-methoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
3-(2-methylpiperidin-1-yl)-N-[2-(trifluoromethoxy)phenyl]azetidine-1-carboxamide
ethyl 1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-5-{[(oxolan-2-ylmethyl)amino]methyl}-1H-pyrazole-4-carboxylate
N-cyclopentyl-4-[2-(2-methoxyethyl)morpholin-4-yl]-4-oxobutanamide