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1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(morpholin-4-yl)propan-1-one
1-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(2-methoxyphenoxy)ethan-1-one
(2R,3R,6R)-5-ethyl-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine
5-methyl-N-[(3-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-1-propyl-1H-pyrazole-4-carboxamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
3-(3-methoxypropyl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
4-{[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
2-(1-benzofuran-2-yl)-6-methylpyridine-3-carboxamide
7-(morpholin-4-ylmethyl)-4-[2-(1H-pyrazol-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-[(3-methyl-1H-indol-2-yl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
(2S,4S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-(pyrimidin-2-ylsulfanyl)pyrrolidine-2-carboxamide
N3-(cyclohexylmethyl)-4-oxo-N5-[(4-phenyloxan-4-yl)methyl]-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-chloro-5-{[7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
1-{2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]ethyl}-2,3-dihydro-1H-imidazol-2-one
methyl 1-({2-[benzyl(methyl)carbamoyl]imidazo[1,2-a]pyridin-3-yl}methyl)piperidine-4-carboxylate
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-({2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholin-4-yl}methyl)quinolin-4-ol
1-ethyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-3-amine
1-(2-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
N'-(2-ethoxyphenyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}propanediamide
(3S,4R)-3-benzyl-1-(2-hydroxybenzoyl)-4-methylpiperidin-4-ol
2-[1-(2-methoxyethyl)pyrrolidin-3-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{4-[(2,3-difluorophenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
N,N-dimethyl-5-{[(2-methylphenyl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[2-methoxy-6-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
methyl 5-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-5-oxopentanoate
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[4-(methylsulfanyl)benzoyl]pyrrolidin-3-yl]methanol
4-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1,2,5-oxadiazole-3-carboxamide
(2S,4R)-N-ethyl-1-(3-methylbut-2-en-1-yl)-4-(4-propylbenzamido)pyrrolidine-2-carboxamide
N-cyclopropyl-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
8-[2-(phenylsulfanyl)ethyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-(morpholin-4-yl)aniline
N-(2,3-dihydro-1H-inden-2-yl)-4-(piperidin-3-yl)benzamide
2-(2-phenyl-1H-imidazol-1-yl)-1-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}ethan-1-one
1-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-hydroxy-3-(2-methylphenoxy)propan-1-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(3-methylpyridin-4-yl)-4-(5-phenyl-1,2-oxazole-3-carbonyl)-1,4-diazepane
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-4-(1H-imidazol-1-yl)butan-1-one
2-[3-({[cyclopropyl(pyridin-2-yl)methyl](methyl)amino}methyl)phenyl]-5-fluoro-6-methyl-3,4-dihydropyrimidin-4-one
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]acetamide
N-(cyclopropylmethyl)-4-(4-methylphenyl)-5-(pyrimidin-5-yl)pyrimidin-2-amine
5-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-N,N-dimethyl-1,2,4-thiadiazol-3-amine
5-[(6-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-[3-(2,6-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-6-methylpyridine
1-[(1S)-1-cyclohexylethyl]-3-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]urea
2-{5-[(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)methyl]-1-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl}acetamide
1-[2-(dimethylamino)ethyl]-4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one
3-(2-fluorophenyl)-1-(2-methoxyethyl)-3-(2-oxo-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}ethyl)pyrrolidine-2,5-dione