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6-methyl-2-{1-[4-(1H-pyrazol-3-yl)benzoyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
4-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}-1-(4-methylphenyl)piperazin-2-one
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(thiophen-2-ylmethyl)-1H-pyrazole-3-carboxamide
methyl 3-acetamido-1-(oxolan-2-ylmethyl)-5-[(4-phenylbutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(ethylamino)-N-(1-hydroxybutan-2-yl)-N-[(2-methylphenyl)methyl]pyrimidine-5-carboxamide
3-{3-[(3,5-dimethoxyphenyl)methoxy]phenyl}-N-methylpyrazin-2-amine
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-(1,3-thiazole-4-carbonyl)-1,4-diazepane
3-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-1-(2,3-dimethylquinoxalin-6-yl)urea
2-(2-methoxyethyl)-4-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}morpholine
3-[(3R,4S)-1-[(5-methylfuran-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[1-(hydroxymethyl)cyclohexyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
[1-(2-methoxyethyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
1-methyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-3-propyl-1H-pyrazole-5-carboxamide
1,3-dimethyl-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
N-({1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
2-(5-hydroxypyrazine-2-carbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
8-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine
3-cyano-N-(2,4-dichloro-3-methylphenyl)piperidine-1-carboxamide
1-{4-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-ylmethyl]phenyl}ethan-1-one
1-(cyclopropylmethyl)-N-ethyl-5-[2-(1,3-thiazol-4-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-[2-(2,4-difluorophenoxy)propanoyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(2-cyanophenyl)-N-[2-(2-methoxyethoxy)phenyl]piperazine-1-carboxamide
2-methoxy-N-[(5-{[3-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]acetamide
1-[(3,4-dimethylphenyl)methyl]-3-(1-ethyl-1H-imidazol-2-yl)piperidine
(2S,4R)-4-amino-N-ethyl-1-{2-[4-(3-methylphenyl)piperazin-1-yl]acetyl}pyrrolidine-2-carboxamide
(1S,5R)-6-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-1H-imidazole-2-carboxamide
N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-methyl-4-({5-[5-(oxolan-2-yl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
{[5-(2-chloro-4-fluorophenyl)-2-methoxyphenyl]methyl}(methyl)amine
5-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]-2-(thiophen-2-yl)pyrimidine
8-methoxy-4-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
ethyl 4-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}piperazine-1-carboxylate
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
5-[4-(4-oxo-3,4-dihydroquinazolin-6-yl)phenyl]imidazolidine-2,4-dione
2-ethoxy-6-{[(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}phenol
N-methyl-3-{[1-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)ethyl]sulfamoyl}benzamide
4-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
6-(methoxymethyl)-2-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
1-benzyl-5-(1-methyl-1H-pyrazole-5-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(3-acetylphenoxymethyl)-N-[(4-fluorophenyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-ylmethyl)acetamide
N-(1-{4-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)oxolane-3-carboxamide
1-[(3-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]-4-methylpiperidine-4-carbonitrile
N-[(2,3-dimethoxyphenyl)methyl]-5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
5-(azepan-1-yl)-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}-4-(naphthalen-1-ylmethyl)piperazin-2-one
1-[(2,3-dimethoxyphenyl)methyl]-3-methylimidazolidin-2-one