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2-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane
4-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-N,N,5,6-tetramethylpyrimidin-2-amine
[(2S)-1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
4-{4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-9H-purin-6-amine
N-(cyclopent-3-en-1-yl)-2-[4-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)morpholin-3-yl]acetamide
1-[4-(morpholin-4-yl)benzoyl]-N-phenylpiperidin-3-amine
N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
1-[4-(dimethylamino)azepan-1-yl]-2-[(2-methylphenyl)sulfanyl]ethan-1-one
(4aS,8aR)-1-butyl-6-(4-methylpiperazine-1-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-{2-[4-(piperidin-1-yl)piperidin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
1-(2-cyclopropylphenyl)-3-[2-(1-methylpyrrolidin-2-yl)ethyl]urea
6-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-9H-purine
1-[(5-methylfuran-2-yl)methyl]-4-oxo-N3-(prop-2-en-1-yl)-N5-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1H-indole
2-(3,5-dimethyl-4-{2-[(3-methylphenyl)carbamoyl]acetamido}-1H-pyrazol-1-yl)acetic acid
1-benzyl-8-[(4-hydroxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(3,5-dimethoxybenzoyl)piperidine-3-carboxylate
3-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1,3-oxazolidin-2-one
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
2-[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]-N-(1,3-thiazol-2-yl)propanamide
2-(dimethylamino)-1-[1-(hydroxymethyl)-9-(pyridin-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
(4aR,7aS)-1-(pyridin-3-ylmethyl)-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 3,5-dimethyl-4-[4-(6-oxo-1,6-dihydropyrimidin-4-yl)piperidine-1-carbonyl]-1H-pyrrole-2-carboxylate
1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-4-phenoxypiperidine-4-carboxylic acid
1-(4-benzylpiperazin-1-yl)-3-[1-(piperidin-4-yl)piperidin-3-yl]propan-1-one
6-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]pyrazine-2-carboxylic acid
1-{1-[(5-methoxy-1H-indazol-3-yl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
(4aS,8aR)-6-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-benzyl-3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-sulfonamide
N-methyl-2-(methylamino)-N-[1-(1,2-oxazol-3-yl)ethyl]pyridine-4-carboxamide
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-2H-1,3-benzodioxole-5-carboxamide
8-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
ethyl 1-(but-3-enoyl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
3-{4-[3-fluoro-5-(propan-2-yloxy)phenyl]-3,5-dimethyl-1H-pyrazol-1-yl}propanamide
1-{2-[2-(2,3,6-trifluorophenyl)-1H-imidazol-1-yl]ethyl}cyclopentan-1-ol
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-[(2,3-dimethoxyphenyl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-(2-methanesulfonylethyl)-3-[(1-methoxypropan-2-yl)sulfamoyl]benzamide
N-[2-(1H-imidazol-4-yl)ethyl]-4-[(pyridin-2-ylmethyl)sulfamoyl]benzamide
2-cyclopentyl-9-(2-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
4-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-4-(3-methylpyridin-4-yl)piperazine
6-(2-{[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-2-methylpyrimidin-4-ol
3-[N-(propan-2-yl)-1-[3-(trifluoromethyl)-1H-pyrazol-5-yl]formamido]propanamide