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1-(2-aminoethyl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
N'-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N'-methyl-N-propylethanediamide
1-(4-chloro-2-fluorophenyl)-3-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]urea
1-(4-fluorophenyl)-4-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,4-diazepane
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
3-[1-(methoxymethyl)cyclopentyl]-1-[4-(2-oxopyrrolidin-1-yl)phenyl]urea
3-(4-hydroxyphenyl)-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1H-pyrazole-5-carboxamide
N-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
5-{2-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}-3-(propan-2-yl)-1,2,4-oxadiazole
N-[3-({[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)carbamoyl}amino)-4-methylphenyl]-2-methoxyacetamide
N-(2-chlorophenyl)-4-(hydroxymethyl)-4-(oxan-2-ylmethyl)piperidine-1-carboxamide
N-[2-hydroxy-2-(3-phenoxyphenyl)ethyl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(3R,4S)-4-(propan-2-yl)-1-(pyrrolidine-1-sulfonyl)pyrrolidin-3-yl]pyrimidin-2-amine
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
2-(2-{[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-[4-({3-[3-(2-methylpyrimidin-4-yl)phenyl]-1H-pyrazol-1-yl}methyl)thiophen-2-yl]ethan-1-one
(1R,5R)-3-benzoyl-6-[(2-ethylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine
5-{[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]methyl}-N-propylpyrimidin-2-amine
2-(4-{1-[(3-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)ethan-1-ol
5-(2,6-difluorophenoxymethyl)-N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
(1S,5R)-6-benzyl-3-[(3,5-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}-4-ethylpiperazine
4-benzyl-1-(5-fluoropentyl)pyrrolidin-2-one
N,N-dimethyl-2-{[methyl({[3-(methylsulfanyl)phenyl]methyl})amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-({4-[6-(propan-2-yl)pyridin-2-yl]piperazin-1-yl}methyl)benzoic acid
N-benzyl{[2-(pyridin-2-ylmethoxy)phenyl]amino}sulfonamide
N4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,4-diamine
4-(3-tert-butyl-5-methylphenyl)-6-(methoxymethyl)pyrimidine
1-(3,4-dimethoxyphenyl)-3-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)urea
2-{1-[2-(3-methoxyphenyl)ethyl]-1H-imidazol-2-yl}pyridine
1-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-(2-methoxyphenoxy)piperidine
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
(3R,4R)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
6-chloro-2-methyl-N-(1,2-oxazol-3-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide
N-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-3-phenylpiperidine-1-carboxamide
methyl[(1-methyl-1H-imidazol-2-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
4-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]thiomorpholine
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-(4-fluorophenyl)-N-[2-(piperidin-1-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
(2S,4S)-4-amino-1-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)acetamide
(3S,4R)-4-(2-methylphenyl)-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]pyrrolidine-3-carboxylic acid
4-[(dimethylamino)methyl]-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)azepan-4-ol
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane