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ethyl 4-{6-[4-(4-fluorophenyl)-4-oxobutanoyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
2-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
methyl 3-{3-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanamido}thiophene-2-carboxylate
1-(5-chlorothiophene-2-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-3-(1H-pyrazol-4-yl)propan-1-one
2-[(5-acetylthiophen-3-yl)methyl]-5-[methyl(2-phenylethyl)amino]-2,3-dihydropyridazin-3-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-3-[(3S,4R)-1-(2-methylpropyl)-4-(morpholin-4-yl)piperidin-3-yl]propanamide
1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}azetidin-3-amine
7-[(3,4-difluorophenyl)methyl]-2-(3-methylpyrazin-2-yl)-2,7-diazaspiro[4.5]decane
N3-[2-(3-chlorophenyl)ethyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{2-[7-(naphthalen-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}oxolane-2-carboxamide
2-methyl-5-{2-[4-(1H-pyrazol-5-yl)phenyl]phenyl}-1,3,4-oxadiazole
1-[3-(3-ethylphenoxy)azetidin-1-yl]-3-(morpholin-4-yl)butan-1-one
(4aR,8aR)-7-[2-(benzyloxy)ethyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-3-(2-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
2-butoxy-1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}ethan-1-one
1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-N-methylpiperidine-2-carboxamide
N-(2-fluorophenyl)-3-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}propanamide
({5-[1-(4-cyclopentylpyrimidin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
[4-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
3-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-1-(3-chloro-4-ethoxyphenyl)-3-methylurea
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-methyl-8-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl 5-{[(4-fluorophenyl)methyl]amino}-1-(2-methoxyethyl)-3-(3-methylbutanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4,4,4-trifluoro-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)butan-1-one
3-{4-[2-(4-fluorophenyl)azetidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
6-tert-butyl-2-{2-[(3,3-dimethylpyrrolidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
1-[3-fluoro-5-(trifluoromethyl)phenyl]-3-(2-hydroxyethyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
2-methyl-4-[3-(2-propylpyrrolidine-1-carbonyl)phenyl]butan-2-ol
2-{4-[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperazin-1-yl}ethan-1-ol
6-(1-benzothiophen-2-yl)-N-benzyl-N-methyl-2-(morpholin-4-yl)pyridine-3-carboxamide
1-(1,4-dithiepan-6-yl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-(4-chlorophenyl)-N-{[1-(pyridin-4-ylmethyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
4-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
3-(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
(3S,4R)-1-(1,4-dithiepan-6-yl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-[2-(dimethylsulfamoyl)ethyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
1-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
1-{4-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-4-oxobutyl}pyrrolidin-2-one
(2,1,3-benzothiadiazol-5-ylmethyl)({[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
4-methyl-6-(propan-2-yl)-2-{4-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]piperidin-1-yl}quinazoline
N-methyl-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidine-2-carboxamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-(phenylamino)pyrimidine-5-carboxamide
3-(benzyloxy)-1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
N,N-dipropyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
N-[(4-hydroxyazepan-4-yl)methyl]-5-(1,2-oxazol-3-yl)thiophene-2-sulfonamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide