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{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[(4-phenyl-1,3-thiazol-5-yl)methyl]amine
3-{5-[2-(propan-2-ylsulfanyl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
methyl 5-({[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}amino)-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3S,4S)-3-hydroxy-N,N-dimethyl-4-(naphthalen-2-yl)piperidine-1-sulfonamide
N-{4-methyl-2-[4-(pyrrolidin-1-yl)butanamido]phenyl}pentanamide
N-(1,4-dioxan-2-ylmethyl)-N,1-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-fluoro-N-methyl-2-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-amine
2-[2-(2-methoxy-4-methylphenoxy)ethyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
N-[2-(2-fluorophenyl)-1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylthiophene-2-carboxamide
N-methyl-3-(2-methylphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)-N-(1,3-thiazol-2-ylmethyl)benzamide
N-(1-benzylpyrrolidin-3-yl)-3-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}propanamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperidine
1-cyano-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
5-(3-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-oxopropyl)-5-[(4-methylphenyl)methyl]pyrrolidin-2-one
3-({3-[5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)-4H-chromen-4-one
(4aS,7aR)-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N2-benzyl-N2,7,7-trimethyl-N5-(piperidin-4-yl)-5,6,7,8-tetrahydroquinazoline-2,5-diamine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(2-hydroxyacetyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,9aR)-8-benzoyl-3-[(1R)-1-(benzyloxy)ethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3R)-3-hydroxy-3,4,4-trimethyl-N-(2-phenylethyl)pyrrolidine-1-carboxamide
[(4-methoxyphenyl)methyl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
2-{[5-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-6-methylpyridine
3-benzyl-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-2-one
1-[(2,6-difluorophenyl)methyl]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
3-(morpholine-4-carbonyl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aS,8aR)-1-(2-phenylethyl)-6-[2-(propan-2-yloxy)acetyl]-decahydro-1,6-naphthyridin-2-one
2-{[(3R,4S)-1-[2-(morpholin-4-yl)-2-oxoethyl]-4-(propan-2-yl)pyrrolidin-3-yl]amino}pyridine-3-carbonitrile
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
2-(dimethylamino)-1-[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]-2-(2-fluorophenyl)ethan-1-one
2-acetamido-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
3-{3-[benzyl(methyl)amino]piperidin-1-yl}-2,2-dimethylpropan-1-ol
(2R,3R,6R)-3-(4-fluorophenyl)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
1-benzyl-5-(pyridine-4-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[1-(3,4-dimethoxyphenyl)-1H-imidazol-2-yl]benzonitrile
1,2-dimethyl-3-(thiomorpholine-4-carbonyl)-1H-indol-5-ol
3-methoxy-1-(2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
N-[4-(3-fluorophenyl)phenyl]-1-(1,3-thiazol-2-yl)piperidine-3-carboxamide
N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
2-(4-chloro-1H-indole-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(furan-2-yl)-3-phenylpropyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
5-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-1H-imidazole-4-carboxylic acid
(3-{2-[1-(4-chloro-2-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-(2-methoxyethyl)-4-oxo-N-[(1-phenylcyclopentyl)methyl]-5-(thiomorpholine-4-carbonyl)-1,4-dihydropyridine-3-carboxamide
5-cyclobutyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1,3,4-oxadiazol-2-amine
N-(butan-2-yl)-3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-[(2-{cyclopropyl[(3-methylthiophen-2-yl)methyl]carbamoyl}phenyl)amino]acetic acid
3-phenyl-N-[4-(4-{[1-(pyridin-3-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]propanamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine