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(2R,3R,6R)-3-(3-methoxyphenyl)-5-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-5-phenyl-1,2-oxazole-3-carboxamide
1-[(3-methoxyphenyl)methyl]-4-(1-methyl-1H-indole-4-carbonyl)piperazin-2-one
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
(3S,9aR)-8-(3-methylbutyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(cyclobutylmethyl)pyrrolidine-3-carboxylic acid
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-cyclopentyl-N-[(3R,4S)-4-cyclopropyl-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]acetamide
(2S,4R)-4-[(4-ethylcyclohexyl)amino]-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-(4-fluorophenyl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]cyclopropane-1-carboxamide
3-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
4,4,4-trifluoro-N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
1-[1-(2-phenylethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-methyl-2-(pyridin-3-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]acetamide
2-(3-chloro-4-hydroxyphenyl)-1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]ethan-1-one
N-(3-chloro-4-methylphenyl)-4-hydroxy-4-(hydroxymethyl)azepane-1-carboxamide
2-(4-methoxyphenyl)-N-({1-[2-(2-oxopiperidin-1-yl)acetyl]piperidin-3-yl}methyl)acetamide
N-[4-(furan-2-yl)butan-2-yl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
6-[4-(1H-imidazol-2-yl)piperidin-1-yl]pyridine-2-carbonitrile
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
2-amino-6-(2,5-dimethoxyphenyl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
1-{9-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl}-2-(methylsulfanyl)ethan-1-one
6-methyl-2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,3-benzodiazole
2-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
1-(4-methoxyphenyl)-2,2-dimethyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]piperazine
2-(pyridin-2-ylmethyl)-8-(pyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-{2-[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-methoxybenzamide
4-(2-{4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazin-1-yl}ethyl)morpholine
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
3-[(2R,3R,6R)-5-[(3-fluoro-4-methylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-{4-[5-(methoxymethyl)thiophene-2-carbonyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
1-[2-(4-chlorophenyl)morpholin-4-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-{4-[(1S,5S)-3,6-diazabicyclo[3.2.2]nonan-3-ylmethyl]thiophen-2-yl}ethan-1-one
2-{1-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
N-{1-[1-benzyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
(1R,3S)-3-(2-aminoethoxy)-7-(furan-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol
1-[(3-methylpyridin-2-yl)methyl]-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazine
2-amino-3-ethyl-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N,N-dimethyl-3-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
3-benzyl-8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-ethyl-1-methyl-3-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-amino-6-cyclobutyl-4-[4-methoxy-3-(methoxymethyl)phenyl]pyridine-3-carbonitrile
1-{3-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenyl}ethan-1-one
N-[4-(5-acetylthiophen-2-yl)phenyl]methanesulfonamide
4-phenyl-2-[4-(pyrrolidine-3-carbonyl)piperazin-1-yl]pyrimidine
4-[(2-ethyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]-N-(1,2,3-thiadiazol-5-yl)benzamide
(3S,4S)-4-cyclopropyl-1-[3-(3-methoxyphenoxy)propyl]pyrrolidine-3-carboxylic acid