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2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-1H-indole
1-[(2-ethylphenyl)methyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
3-(difluoromethoxy)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
1-(benzenesulfonyl)-4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazine
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)oxane-4-carboxamide
4-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-2-(2-phenylethyl)morpholine
9-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-3-azaspiro[5.5]undecane
1-[1-(6-aminopyrimidin-4-yl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
4-(pyrrolidine-1-carbonyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzene-1-sulfonamide
2-[4-methyl-1-(pyridin-4-yl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
2-[4-(1H-pyrazol-3-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
N-(oxolan-3-ylmethyl)-3-(pyridin-2-yl)-1H-pyrazol-5-amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-5-(methoxymethyl)-N-methylfuran-2-carboxamide
3-{4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-5-methylpyridine
3-ethyl-8-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(2-methoxyphenoxy)-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}azetidine
2-cyclopentyl-N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]acetamide
3-[(3R,4S)-1-(5-chlorothiophene-2-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-{2-[(2R)-2-amino-3-hydroxypropanamido]-4-methylphenyl}benzamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
N-[2-(2,4-dimethoxyphenyl)ethyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-2,3-dihydro-1H-isoindole
methyl 6-[({2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}carbamoyl)amino]-1,2,3,4-tetrahydroquinoline-1-carboxylate
3-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-1H-indazole
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
3-[(1-benzylpyrrolidin-3-yl)amino]-N-(furan-2-ylmethyl)propanamide
5-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[(4-fluorophenyl)methyl]-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
(4S)-3-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-6-(3-methoxyphenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
2-methyl-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}pyrimidin-4-ol
1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-7-oxoazepan-4-yl}-N,N-diethylpiperidine-3-carboxamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-[(1-methylpyrrolidin-2-yl)methyl]-1,3-oxazole-4-carboxamide
(3S,7S)-5-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
5-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
1-(4-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
5-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
3-(2-fluorophenyl)-1-(2-methoxyethyl)-3-{2-oxo-2-[3-(2-phenylacetyl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
1-(1H-imidazol-2-ylmethyl)-4-(2-methoxyethyl)piperidine-4-carboxylic acid
2,6-difluoro-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
5-butyl-1'-(1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[4-(5-chloro-2-methylphenyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-3-(oxolan-3-yl)-1-phenyl-1H-1,2,4-triazole
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-(4-{2-[2-(3-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)propan-1-one
2-{2-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one