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N-cyclopentyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-1,3-thiazole-5-carboxamide
2-methyl-6-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]pyrimidin-4-amine
1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-3-methylbut-2-en-1-one
1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-sulfamoylbenzamide
1-butyl-5-({8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-2-(ethanesulfonyl)-1H-imidazole
N-[(3,4-dimethoxyphenyl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
4-(4-phenyl-1H-pyrazol-5-yl)-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
3-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-(oxolan-3-ylmethyl)piperidine
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-4-(thiophen-2-yl)butan-1-one
5-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
(3aR,5S,6S,7aS)-2-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-octahydro-1H-isoindole-5,6-diol
3-[4-(1H-imidazol-1-yl)phenyl]-1-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}urea
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-3-phenyl-1H-pyrazole-5-carboxamide
3-({[1-(5-chloro-2-methoxybenzoyl)piperidin-4-yl]oxy}methyl)pyridine
(1S,6R)-9-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(3S,7S,8aS)-7-({[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}amino)-3-propyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
5-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-(3-fluorophenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
ethyl 4-{2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
4-({4-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}methyl)thiomorpholine
N-[3-(1H-indol-2-yl)phenyl]-1-propanoylpiperidine-3-carboxamide
5-(morpholin-4-ylmethyl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}furan-3-carboxamide
1-phenyl-4-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperazine
2-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4-methyl-1H-imidazole
methyl 4-({methyl[(1-phenylpyrrolidin-3-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylate
(2R,6S)-2,6-dimethyl-4-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}morpholine
N-{[1-(isoquinolin-5-ylmethyl)pyrrolidin-3-yl]methyl}-2-methoxyacetamide
4-{2-[4-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
(4aR,8aR)-7-(3-cyano-6-methylpyridin-2-yl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
N,N,4-trimethyl-6-(4-{[(5-methyl-1H-pyrazol-3-yl)methyl]amino}piperidin-1-yl)pyrimidin-2-amine
1-(2-{3-[1-(3,3,3-trifluoro-2-hydroxypropyl)-1H-pyrazol-3-yl]phenyl}phenyl)ethan-1-one
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-4-ol
4-{[methyl(2-phenoxyethyl)amino]methyl}benzene-1,2-diol
4-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,N-dimethylbenzamide
2-({[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}(thiophen-2-ylmethyl)amino)butan-1-ol
4-methanesulfonyl-2-{[4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,2,3-triazol-1-yl]methyl}morpholine
1-[(4-chlorophenyl)methyl]-N-methyl-N-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-[1-(2-chloro-4,5-difluorobenzoyl)piperidin-2-yl]pyridine
(2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]pyrrolidine-2-carboxylic acid
2-[1-(2-methoxyethyl)piperidin-4-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-2-(methylamino)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-thiazole-4-carboxamide
4-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-4H-1,2,4-triazole
5-methoxy-9-[4-(pyrrolidin-1-ylmethyl)benzoyl]-1-oxa-9-azaspiro[5.5]undecane
(2,1,3-benzothiadiazol-5-ylmethyl)[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amine
(4aS,8aR)-1-butyl-6-[3-(1,2-oxazinan-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
N-(3-methyl-1H-pyrazol-5-yl)-2-(1-methyl-1H-pyrrol-3-yl)acetamide
1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
N-[(7-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-3-(pyridin-3-yl)propanamide
N-[3-(dimethylamino)propyl]-1-methanesulfonyl-N-methylpiperidin-3-amine