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2-[3-(1H-pyrazol-1-yl)benzoyl]-2,7-diazaspiro[4.5]decane
9-[(2-aminopyridin-3-yl)methyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidin-4-yl)methyl]acetamide
N-[(4-fluorophenyl)methyl]-1-methyl-5-{[2-(pyridin-3-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}-4-(thiophen-2-yl)butan-1-one
N-[(3R,4R)-1-[3-(2-fluorophenyl)propanoyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-methylpiperidine
(2R,3R,6R)-5-(2,4-difluorobenzoyl)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-{[2-methyl-5-(trifluoromethyl)phenyl]methyl}-1,3-oxazolidin-2-one
2-(6-methylpyridazin-3-yl)-2,7-diazaspiro[4.5]decane
N-[(3R,4S)-4-cyclopropyl-1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]pyrrolidin-3-yl]acetamide
N,N-diethyl-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carboxamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(2-methoxyacetyl)-decahydro-1,6-naphthyridin-2-one
3,4-difluoro-N-{[1-(pyrimidin-2-ylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}benzamide
1-[4-(furan-3-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
2-ethyl-N-[2-(pyridin-3-yl)ethyl]pyrimidine-5-carboxamide
2-(2-methoxy-5-methylphenyl)-2-[methyl(2-methylprop-2-en-1-yl)amino]acetic acid
9-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(1H-pyrazol-1-yl)propyl]propanamide
N-[(2S)-2-aminopropyl]-2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzamide
ethyl 4-(1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1H-pyrazol-4-yl)propanamide
3-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-N-(3-chloro-4-methoxyphenyl)propanamide
1-[1-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)azetidin-3-yl]-2-methylpiperidine
1-methyl-9-[4-(1H-pyrazol-5-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
(1S,2S)-2-{4-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-1-yl}cyclohexan-1-ol
1-(1H-1,3-benzodiazol-5-yl)-3-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)urea
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl}propanamide
1,6-dimethyl-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[2-(ethylamino)pyrimidine-5-carbonyl]-N,N-dimethylpiperazine-1-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-indazol-1-yl)propyl]acetamide
(3-{[(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amino]methyl}-2,4,6-trimethylphenyl)methanol
3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]pyridin-2-ol
4-[(2-phenyl-1H-imidazol-4-yl)methyl]-1,4-oxazepane
2-[1-(2-fluorophenyl)piperidin-4-yl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-3-(quinolin-8-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[4-(1H-indazole-3-carbonyl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
N-{2-[5-(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
methyl (2S,4R)-1-(3-phenylpropyl)-4-(thiophene-2-amido)pyrrolidine-2-carboxylate
1-(1-methylazepane-2-carbonyl)-4-phenyl-1,4-diazepane
1-(dimethylamino)-2-{4-[(3-ethoxy-4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
N-[2-(pyridin-3-yloxy)phenyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-phenylpropyl)acetamide
1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-3-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}urea
(3S,4R)-1-(5-chloro-3-fluoropyridin-2-yl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
(2E)-1-{4-[2-(naphthalen-1-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
2-[2-(4-chlorophenyl)morpholin-4-yl]-N,N-diethylacetamide