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N-(3-cyanophenyl)-5-{1-[(5-methylfuran-2-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-chloro-2-propanamido-N-[4-(1H-pyrazol-1-yl)butan-2-yl]benzamide
N-butyl-1-(difluoromethyl)-N-[(3-methoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
8-(1-acetylpiperidine-4-carbonyl)-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[(5-methylpyrazin-2-yl)methyl]propanamide
1-(diethylamino)-3-[4-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,4-dimethylbenzamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
[(2S,6S)-4-(2,3-difluoro-6-methoxybenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-(2-methylpropyl)piperidine-3-carboxamide
4-{4-[2-(2-fluorophenyl)acetyl]piperazin-1-yl}-2-[2-(4-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
N-(3-chloro-2-methylphenyl)-N'-[2-(pyridin-2-yl)ethyl]propanediamide
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
N-[(4-hydroxyphenyl)methyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
3-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-2-(methylsulfanyl)pyridine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-7-oxo-2-(2-phenylacetamido)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-ethyl-N-methyl-2-oxo-N-[(4-phenoxyphenyl)methyl]-1,2-dihydropyridine-4-carboxamide
(2R,6R)-4-[(3,4-dimethoxyphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{4-[(4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenyl}acetamide
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-{[2-(methylsulfanyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-methoxy-1-[1'-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-4-[(4-methylphenyl)methyl]-1,4-diazepan-5-one
3-(2-methoxyphenyl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]propanamide
2-(3-methylphenyl)-5-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)pyrimidine
N-{1-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-1,2-oxazole-5-carboxamide
1-(3-{3-[(4-benzylpiperidin-1-yl)methyl]phenoxymethyl}piperidin-1-yl)propan-1-one
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-[(3-ethoxy-4-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
N-cyclobutyl-3-{[2-(ethylsulfanyl)ethyl]sulfamoyl}benzamide
1-(4-fluorophenyl)-5-[1-(methoxymethyl)cyclobutyl]-3-methyl-1H-1,2,4-triazole
ethyl 2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
3-(4-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}phenyl)-1H-1,2,4-triazole
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(dimethylamino)benzamide
ethyl 1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
4-{4-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]piperidin-1-yl}-N-(pyridin-3-ylmethyl)benzamide
[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)propylamine
(1R,3R)-N1-(3,5-dichloropyridin-2-yl)cyclopentane-1,3-diamine
N,N-diethyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
2-methoxy-1-[1'-(1,3-thiazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
4-(4-fluorophenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}oxane-4-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)cyclopropanecarboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2,6-dimethylpyridine-4-carboxamide
2-{4-[2-(dimethylamino)ethoxy]piperidin-1-yl}-2-[4-(methylsulfanyl)phenyl]acetic acid
5-{3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2-ethylpyrimidine