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1-(azepan-1-yl)-3-[2-methoxy-4-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-methoxy-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine
1-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
({1-ethyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}(3-fluorophenyl)methyl)dimethylamine
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-{4-[(3-{[1-(5-chloro-2-methoxybenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]piperazin-1-yl}pyrimidine
1-[2-(dimethylamino)ethyl]-3-(2-methylphenyl)-3-{2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
1-{4-[2-(phenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
3-methyl-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-1-propyl-1H-pyrazole-4-carboxamide
3-(4-{[2-(propylamino)pyrimidin-5-yl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile
N-[(3S,4R)-1-[(6-fluoroquinolin-2-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
1-methyl-N-(thiophen-2-ylmethyl)-5-[(2,2,2-trifluoroethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2-ethoxyphenyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
2-(3-chlorophenyl)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-hydroxyethan-1-one
(1S,5R)-6-benzyl-3-{[2-(methylsulfanyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl (2S,4R)-1-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-4-(dimethylamino)pyrrolidine-2-carboxylate
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(2,5-difluorophenyl)methyl]pyrrolidin-3-yl]methanol
2-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}phenol
3-{methyl[2-(pyridin-2-yl)ethyl]amino}-N-(4-phenoxyphenyl)piperidine-1-carboxamide
2-methyl-N-(morpholin-2-ylmethyl)-1-benzofuran-5-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2,6-dimethylquinoline-4-carboxamide
1-(9-{[2-(ethylamino)pyrimidin-5-yl]methyl}-3,9-diazaspiro[5.5]undecan-3-yl)-2-methoxyethan-1-one
(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperidin-3-yl)methanamine
N-[(8-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]acetamide
8-(pyridin-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}morpholine
1-(2-methylpropyl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(2-oxopyrrolidin-1-yl)propanamide
3,4,7-trimethyl-2-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-1H-indole
2-methyl-6-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)pyridine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]azetidine-1-carboxamide
1-(3-methylpyridin-2-yl)-4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperazine
1-[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(furan-2-yl)propan-1-one
(3aS,6aS)-2-(ethanesulfonyl)-5-(3-fluoropyridin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 4-{12-oxo-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-14-yl}-1H-pyrazole-3-carboxylate
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-(3-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(4-phenylpiperidin-1-yl)acetamide
N-{[7-(5-acetylthiophene-3-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
3-{3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-methylpyridine
6-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-amine
4-{1-[4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)phenyl]ethyl}morpholine
dimethyl({4-methyl-5-[1-(pyridin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(1-methyl-1H-pyrazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-(1-{[(2-butoxy-3-methoxyphenyl)methyl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-fluorophenyl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
N-[(3S,4R)-1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-2-(2-propyl-1H-1,3-benzodiazol-1-yl)propanamide
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-[2-(hydroxymethyl)pyridin-4-yl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1,4-diazepan-5-one
4-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyrimidin-2-yl)morpholine