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[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl][3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amine
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
8-({2-[(carboxymethyl)(methyl)amino]pyrimidin-5-yl}methyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3S,4S)-3-hydroxy-4-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-1λ6-thiolane-1,1-dione
3-ethyl-6-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
[3-(prop-2-en-1-yl)-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl]methanol
(2S,4R)-4-[(adamantan-2-yl)amino]-1-[(2-chlorophenyl)methyl]-N,N-diethylpyrrolidine-2-carboxamide
6-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
8-(4-hydroxybenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
[(4aS,8aR)-6-[2-(morpholin-4-yl)benzoyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
6-(1-{2-oxo-1-oxaspiro[4.4]nonane-4-carbonyl}piperidin-3-yl)-3,4-dihydropyrimidin-4-one
ethyl 6-[4-(oxan-4-yl)piperazin-1-yl]pyridine-3-carboxylate
(2S,4R)-1-benzyl-N-methyl-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-ethyl-N-[(4-methoxyphenyl)methyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-{3-[6-amino-5-cyano-4-(furan-2-yl)pyridin-2-yl]-1H-indol-1-yl}propanoic acid
4-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-1,2-dihydroquinazolin-2-one
methyl 2-[3-(4-methoxyphenyl)-N-methyl-3-phenylpropanamido]acetate
(2R,3R,6R)-5-[(2,3-difluorophenyl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-3-(pyrimidin-2-yloxy)benzamide
N-(2-{7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
1-[(3-chlorophenyl)methyl]-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-phenylcyclopropyl)acetamide
2-(5-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}furan-2-yl)benzonitrile
(1S,4S)-2-[2-(methylsulfanyl)phenyl]-5-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
6-methyl-3-[2-(morpholin-4-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
7-fluoro-3-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-1-[2-(phenylsulfanyl)ethyl]-1,2-dihydroquinolin-2-one
4-(propan-2-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}pyrimidin-2-amine
1-ethyl-5-(1-{[4-(trifluoromethyl)phenyl]methyl}-1H-imidazol-2-yl)-1H-1,2,4-triazole
methyl 4-({4-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}methyl)benzoate
N-[(2R,3R)-1'-[(2,6-dimethoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
N-({7-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenoxypropanamide
6-[2-(1-benzylpiperidin-2-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-(2-methylpropyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-5-carboxamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methoxyphenyl)acetamide
N-cyclopropyl-1-{1-[(4-fluoro-3-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-[(3R,4S)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
ethyl 1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
2-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
9-(5-acetylpyridin-2-yl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]pyrrolidin-2-one
N5-[(5-chlorothiophen-2-yl)methyl]-N6-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)propanamide
methyl 3-(2,4-dimethylbenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
7-(3-chlorophenyl)-4-(1-methyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[(3,4-difluorophenyl)methyl]-N-ethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
methyl 5-[2-(6-methyl-1-benzofuran-3-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
(4aR,8aS)-1-butyl-6-{[5-(methoxymethyl)furan-2-yl]methyl}-decahydro-1,6-naphthyridin-2-one
4-{5-[(2-fluoro-4-methoxyphenyl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[phenyl(pyridin-4-yl)methyl]-1H-pyrazole-4-carboxamide