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3-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
(furan-3-ylmethyl)({[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl})amine
methyl 3-acetamido-5-{[(3-fluorophenyl)methyl]amino}-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[(4-cyclopropyl-5-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)(prop-2-yn-1-yl)amine
N-(2,3-dihydro-1H-inden-2-yl)-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-methyl-1-phenyl-5-[3-(1H-pyrazol-3-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2,2-dimethyloxan-4-yl)benzamide
(3aR,6aS)-5-[3-(dimethylcarbamoyl)pyridin-2-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(6-hydroxy-1,4-oxazepan-4-yl)-6-(trifluoromethyl)pyridine-3-carboxamide
2-methyl-5-{[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]methyl}pyrazine
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2,4-dimethyl-1,3-thiazole-5-carboxamide
3-[(4-{[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]amino}-6-methylpyrimidin-2-yl)amino]phenol
1-[4-(piperidin-1-ylmethyl)benzoyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]-1,4-diazepan-5-one
4-(2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)piperazin-2-one
1-methyl-2-oxo-6-(propan-2-yl)-N-[(3,4,5-trimethoxyphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(thiophen-2-ylmethyl)benzamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methoxybenzamide
1-(4-fluoro-3-methoxyphenyl)-3-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}urea
ethyl 2-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-2-yl)acetate
6-oxo-1-(3-phenylpropyl)-N-[4-(pyridin-2-yl)butyl]piperidine-3-carboxamide
N-{2-[(4-fluorophenyl)formamido]ethyl}-2-(propan-2-yloxy)propanamide
3-{1-[(2,5-difluorophenyl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
2-[({[3-(ethoxymethyl)-4-methoxyphenyl]methyl}(methyl)amino)methyl]-3,4-dihydroquinazolin-4-one
methyl 4-[3-(2-{methyl[2-(pyridin-2-yl)ethyl]carbamoyl}ethyl)piperidin-1-yl]-4-oxobutanoate
6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,3-benzothiazole
2-(cyclohex-1-en-1-yl)-1-{4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-4-methyl-1,3-oxazole-5-carboxamide
N-(1-hydroxybutan-2-yl)-5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)pyridazine-3-carboxamide
methyl 6-(2-cyclopropylacetyl)-2-[(4-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3R,4R)-4-methyl-3-(propan-2-yl)-1-{2-[(propan-2-yl)amino]pyrimidine-5-carbonyl}pyrrolidin-3-ol
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
3,4,7-trimethyl-2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}-1H-indole
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(methylsulfanyl)propan-1-one
2-methoxy-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
2-cyclopentyl-N-[7-(4-methoxypiperidine-1-carbonyl)-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazol-5-yl]acetamide
5-ethyl-4-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]-2-methylpyrimidine
2-(adamantan-1-yl)-4-hydroxy-N-(1-hydroxybutan-2-yl)pyrimidine-5-carboxamide
7-ethyl-2-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
[1-(2-chlorobenzenesulfonyl)-3-[(3-chlorophenyl)methyl]piperidin-3-yl]methanol
N-(butan-2-yl)-3-(1H-pyrazol-1-ylmethyl)-N-(pyridin-4-ylmethyl)benzamide
2-{3-[3-(2-chlorophenoxy)azetidine-1-carbonyl]phenyl}-1H-imidazole
1-(2-aminoethyl)-N-[1-(benzenesulfonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-{[3-(furan-2-yl)phenyl]methyl}-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
N-[(2-methoxyphenyl)methyl]-2-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-(4-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3-(1-methylpiperidin-3-yl)propanamide
N4,N4,5-trimethyl-N2-[2-(morpholin-4-yl)ethyl]pyrimidine-2,4-diamine