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N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-{4-[(2,3-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-3-methylbutan-1-ol
(1S,9S)-11-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
[3-(2-methoxyethyl)-1-(4-propylpyrimidine-5-carbonyl)piperidin-3-yl]methanol
[3-methyl-1-(2,7,8-trimethylquinoline-4-carbonyl)piperidin-3-yl]methanol
2-(ethoxymethyl)-N-[1-(5-methylpyridin-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2,3,4,9-tetrahydro-1H-carbazole-7-carboxamide
2-methoxy-4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
(3S,4S)-1-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[(3-chloro-1-benzothiophen-2-yl)methyl]amine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
7-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-chlorobenzamide
(2S,4R)-4-{9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-amido}-1-methyl-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-(2-propyl-2,5-dihydro-1H-pyrrol-1-yl)ethan-1-one
3-(methanesulfonylmethyl)-1-[(5-phenylthiophen-2-yl)methyl]piperidine
{1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
1-{2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
7-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-2,3,6-trimethylquinoline-4-carboxamide
1-(3-hydroxyphenyl)-5-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrrolidine-3-carboxamide
5-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]furan-2-carboxylic acid
1-(5-tert-butyl-1,3,4-oxadiazol-2-yl)piperidine-3-carboxamide
N,2-diethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(1S,6R)-9-[5-(trifluoromethyl)pyridin-2-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(4aS,7aR)-4-(2-methoxyethyl)-6,6-dioxo-N-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
6-ethoxy-4-methyl-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]quinazoline
1-benzyl-4-oxo-N-(propan-2-yl)-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
5-amino-3-(3-ethenylphenyl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
3-({1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
1,3-dimethyl-N-[5-(morpholin-4-yl)pentyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
7-(2,4,5-trimethylbenzoyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
2-(dimethylamino)-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}acetamide
3-(2-methylphenyl)-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
methyl 1-[(3R,5S)-1-(2-methylpropyl)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-{4-[2-(3-fluoropyridin-4-yl)-1H-imidazol-1-yl]phenyl}-5-methylfuran-2-carboxamide
6-{pyrazolo[1,5-a]pyridin-7-yl}-1H-indole
[(3R,4R)-1-(1-benzothiophene-2-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-(1-benzoxepine-4-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-[1-(3-methoxypyrazin-2-yl)piperidin-4-yl]pyrrolidin-2-one
3-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
2-(2-hydroxypropyl)-9-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl][(4-fluoro-3-methoxyphenyl)methyl]methylamine
N-{1-[1-(cyclohexylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
2-{2-[3-methyl-4-(propan-2-yl)piperazin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-[(3S,4R)-1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-4-propylpyrrolidin-3-yl]methanesulfonamide
7-[(2,3-dimethoxyphenyl)methyl]-2-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-2,7-diazaspiro[4.5]decane