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N-(2-ethylphenyl)-4-[2-(phenylcarbamoyl)ethyl]piperidine-1-carboxamide
3-[(dimethylamino)methyl]-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-3-ol
4-(pentan-2-yl)-1-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole
(furan-3-ylmethyl)(methyl){[5-(1H-1,2,4-triazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine
3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
1-[3-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenyl]ethan-1-one
6-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1H-indole
N-methyl-2-(3-phenylpropyl)-N-(pyrazin-2-ylmethyl)-1,3-benzoxazole-5-carboxamide
5-(3-methoxyphenoxymethyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
2-{4-[1-(2-fluorophenyl)piperidin-4-yl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-ethyl-5-methyl-6-[4-(thian-4-yl)piperazin-1-yl]pyrimidin-2-amine
3-(2-chlorophenyl)-3-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}propanamide
1-methyl-6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
2-methoxy-N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-2H-1,3-benzodioxole-5-carboxamide
1-[3-(4-methylphenoxymethyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-ylmethyl)piperidine
N4-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-6-(propan-2-yl)pyrimidine-2,4-diamine
4-ethyl-3-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}naphthalene-1-carboxamide
4-chloro-1-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H-pyrazole-3-carboxamide
methyl({[2-(propan-2-yl)pyrimidin-4-yl]methyl}){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
2-({4-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
2-(3-fluoro-4-methoxyphenyl)-2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}acetic acid
2-{2-[2-(4-fluorophenoxy)ethyl]phenyl}-5-methyl-1,3,4-oxadiazole
1-[1-(azepane-1-sulfonyl)-4-phenylpiperidin-4-yl]ethan-1-one
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(1-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[2-(difluoromethoxy)benzoyl]-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
5-methanesulfonyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
2-ethyl-6-(2-methyl-1-benzofuran-7-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-(2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)piperidine-3-carboxamide
2-(butylsulfanyl)-N4-[(1-methanesulfonylpiperidin-3-yl)methyl]pyrimidine-4,6-diamine
9-[(dimethyl-1,3-thiazol-5-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(3R,5S)-N3-(3-methoxypropyl)-N5-(4-methylphenyl)piperidine-3,5-dicarboxamide
2-[(4-fluorophenyl)methyl]-4-(oxan-4-yl)morpholine
N-[2-(3-phenylpiperidin-1-yl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methylacetamide
1-ethyl-4-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[4-(2-fluorophenyl)benzoyl]-1,4-diazepan-5-one
N-cyclohexyl-N-methyl-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(1,2-oxazinan-2-yl)propanamide
2-methyl-5-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1H-1,3-benzodiazole
2-{2,7-diazaspiro[4.5]decan-2-yl}pyridine-4-carboxamide
N-(2-hydroxy-2-phenylethyl)-N,5-dimethyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
7-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-2-methyl-2,7-diazaspiro[4.5]decane
N,1-dimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
N-[(4-fluoro-2-methylphenyl)methyl]-1-methyl-N-(pyridin-3-ylmethyl)piperidin-4-amine