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2-(3-methoxypropyl)-4-[3-(piperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
ethyl 3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
ethyl 4-[3-({[2-(3-fluorophenyl)ethyl]amino}methyl)-6-methylquinolin-2-yl]piperazine-1-carboxylate
N-methyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
6-[4-(3-methylphenoxy)piperidin-1-yl]pyrimidin-4-amine
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-(2-oxo-2-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}ethyl)-1,4-dihydroquinolin-4-one
N'-(3-chloro-4-methylphenyl)-N-methyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}propanediamide
2-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetic acid
{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-({7-[3-(2-methoxyphenyl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(piperidin-1-yl)acetamide
N,1,3,5-tetramethyl-N-[1-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-methyl-3-phenylpiperidine
1-cyclopentyl-N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-6-oxopiperidine-3-carboxamide
2-(3-benzyl-1,2,4-oxadiazol-5-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-(thiophene-3-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N,N-dimethylpiperidine-4-carboxamide
N-cyclopropyl-2-{[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]oxy}-4-methoxybenzamide
9-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1,4,9-triazaspiro[5.5]undecan-5-one
2-{1-[4-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-imidazol-2-yl}pyridine
N-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-2-(1H-imidazol-2-yl)benzamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
[1-(morpholine-4-sulfonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
N3-tert-butyl-4-oxo-1-(propan-2-yl)-N5-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3,5-dicarboxamide
2-[2-(3-fluoro-4-methoxybenzoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
2-amino-4-{3-[2-(dimethylamino)ethoxy]phenyl}-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
(3aR,6aS)-1-oxo-5-[6-(trifluoromethyl)pyridin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-[(2-oxo-1,2-dihydropyridin-1-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
N-methyl-N-[(5-methylfuran-2-yl)methyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
4-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-1,2-dihydrophthalazin-1-one
3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-N-cycloheptylpiperidine-1-carboxamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[(4-methanesulfonylphenyl)methyl]methylamine
6-methyl-N4-[(2,4,5-trifluorophenyl)methyl]pyrimidine-2,4-diamine
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazol-3-yl]acetamide
1-{1H-pyrrolo[2,3-b]pyridin-6-yl}-3-(thiophene-2-carbonyl)piperidine
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({[1-(phenoxymethyl)cyclopropyl]methyl})amine
(3S)-N,N-dimethyl-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}azepan-3-amine
methyl 2-(1-{1-[(4-chlorophenyl)methyl]-6-oxopiperidin-3-yl}-N-methylformamido)acetate
6-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-(morpholin-4-yl)pyrimidin-4-amine
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-[(6-methylpyridin-2-yl)methyl]propanamide
2-(4-hydroxyphenyl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
1-(3-fluorophenyl)-3-{1-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
(3aS,7aR)-5-methyl-2-(2-methyl-1,3-thiazole-4-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
[(3R,4S)-1-[(3,5-difluorophenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-(4-methylphthalazin-1-yl)-7-azaspiro[3.5]nonan-1-ol
1-[5-(methoxymethyl)thiophene-2-carbonyl]-3-(3-methoxypropyl)piperidine