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1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(2-methylphenyl)sulfanyl]piperidine
5-methyl-1-(4-methylphenyl)-4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-2-one
2-butyl-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-({5-[(1-ethylpiperidin-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
3-(3-fluorophenyl)-1-methyl-3-[2-(3-methylpiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
2-(4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-2-(2,4-dichlorophenoxy)-N-methylacetamide
3-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
4-(3-hydroxy-3-methylbutyl)-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]benzamide
5-(2-chloro-4-fluorophenoxymethyl)-N-[3-(1H-pyrazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
(3S,4S)-1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
5-acetyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}thiophene-3-carboxamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
N3-[(4-fluorophenyl)methyl]-N1,N1-dimethyl-N3-(prop-2-yn-1-yl)piperidine-1,3-dicarboxamide
6-(3-methoxyphenyl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
[2-(6-methoxynaphthalen-2-yl)phenyl]methanamine
4-[(2R)-2-hydroxy-2-(naphthalen-2-yl)acetyl]piperazine-1-sulfonamide
1-cyclohexyl-4-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
4-(1H-imidazol-1-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]benzamide
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)-3,4-dimethylbenzamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(methylsulfanyl)-N-(oxolan-2-ylmethyl)propanamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-2-methoxy-N-(oxolan-2-ylmethyl)benzamide
N-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridin-2-yl)-2,2-dimethylpropanamide
2-(1,5-dimethyl-1H-indazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(dimethyl-1,2-oxazol-4-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-2-carboxamide
1-methyl-2-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
1-{2-oxo-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,2-dihydropyrimidin-2-one
1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(3-methoxypropyl)piperidine
2-(2,2-dimethylpropyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(4,6-dimethylpyrimidin-2-yl)-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}piperidin-4-amine
[(2S,4R,5R)-5-(4-chlorophenyl)-4-{[({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)amino]methyl}-1-ethyl-2-methylpyrrolidin-2-yl]methanol
2-{[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrol-2-yl]methyl}-6-fluoroquinolin-4-ol
3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)benzene-1-sulfonamide
3,3-dimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]cyclohexan-1-amine
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-methyl-N-[(4-phenoxyphenyl)methyl]propanamide
1-ethyl-5-{[4-(2-phenylethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-1,2,4-triazole
N-(adamantan-1-ylmethyl)-N-(2-hydroxyethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
7-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-{4-[2-amino-3-cyano-6-(2-methylbutan-2-yl)pyridin-4-yl]phenoxy}acetamide
ethyl 1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(cyclopropylmethyl)piperidine-4-carboxylate
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-3-(pyridin-4-yl)propanamide
5-[1-(2-fluorophenyl)-1H-pyrazol-3-yl]-4-methyl-N-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-1,3-thiazol-2-amine
2-phenoxy-1-[2-(thiomorpholin-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
N-methyl-2-[4-(2-oxoimidazolidin-1-yl)phenyl]-N-(quinolin-5-ylmethyl)acetamide
7-(6-fluoro-4-hydroxyquinoline-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(4-hydroxyphenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-methyl-1-{4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}propan-1-one
(3S)-3-({[7-chloro-2-(2-phenylethoxy)quinolin-3-yl]methyl}amino)azepan-2-one